| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3536917 | A | Drug uptake assessed as OCT1 (unknown origin)-mediated drug uptake expressed in HEK293 cells by liquid scintillation counting relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 2. | ALA3536922 | A | Inhibition of OCT1 (unknown origin) expressed in HEK293 cells assessed as reduction of [14C]metformin substrate uptake at 100 uM by liquid scintillation counting | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 3. | ALA3536923 | A | Inhibition of OCT1 (unknown origin) expressed in HEK293 cells assessed as reduction of [ethyl 1-14C]TEA substrate uptake at 100 uM by liquid scintillation counting | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 4. | ALA4809211 | B | Inhibition of human OCT1 assessed as reduction in OCT1-mediated metformin transport at 14900 uM relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 5. | ALA4825999 | B | Inhibition of human OCT1 assessed as reduction in intracellular probe substrate accumulation upto 100 uM by microplate scintillation counter analysis relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 6. | ALA4828793 | B | Substrate activity at human OCT1 expressed in HEK293 cells assessed as increase in compound uptake by measuring Km incubated for 2 mins by LC-MS/MS analysis | Homo sapiens | 22 | cell-based format | Scientific Literature | ||
| 7. | ALA4828794 | B | Substrate activity at human OCT1 expressed in HEK293 cells assessed as increase in compound uptake by measuring Vmax incubated for 2 mins by LC-MS/MS analysis | Homo sapiens | 22 | cell-based format | Scientific Literature | ||
| 8. | ALA4828795 | B | Substrate activity at human OCT1 expressed in HEK293 cells assessed as increase in compound uptake by measuring intrinsic clearance incubated for 2 mins by LC-MS/MS analysis | Homo sapiens | 22 | cell-based format | Scientific Literature | ||
| 9. | ALA4837389 | B | Inhibition of OCT1 (unknown origin) expressed in HEK293 cells | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 10. | ALA5119566 | B | Inhibition of OCT1 (unknown origin) overexpressed in HEK293 cells assessed as intracellular accumulation of ASP+ measured at 20 uM for 5 mins by Analyst AD plate reader method relative to control | Homo sapiens | 8 | cell-based format | Scientific Literature | ||
| 11. | ALA5119570 | A | Substrate activity at human OCT1 overexpressed in HEK293 cells at 2.5 uM incubated for 2 mins by LC-MS/MS analysis | Homo sapiens | 7 | cell-based format | Scientific Literature | ||
| 12. | ALA5119577 | A | Substrate activity at OCT1 (unknown origin) assessed as uptake ratio | Homo sapiens | 6 | cell-based format | Scientific Literature |
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