| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3592404 | B | Inhibition of PRDM9 (unknown origin) assessed as incorporation of tritium labeled methyl group from [3H]-SAM to substrate at 1 uM after 1 hr by scintillation proximity assay relative to control | Homo sapiens | 1 | ALA3588844 | single protein format | Scientific Literature | |
| 2. | ALA3784093 | B | Inhibition of human PRDM9 at 10 and 50 uM | Homo sapiens | 1 | ALA3779843 | single protein format | Scientific Literature | |
| 3. | ALA3803127 | B | Inhibition of PRDM9 (unknown origin) at 10 uM relative to control | Homo sapiens | 2 | ALA3797202 | single protein format | Scientific Literature | |
| 4. | ALA3821563 | B | Inhibition of PRDM9 (unknown origin) at 1 to 50 uM by scintillation proximity assay | Homo sapiens | 1 | ALA3817823 | single protein format | Scientific Literature | |
| 5. | ALA3859066 | B | Inhibition of PRDM9 (unknown origin) at 50 uM using biotin-labeled peptide as substrate and [3H]-SAM measured after 1 hr by scintillation proximity assay | Homo sapiens | 1 | ALA3856251 | single protein format | Scientific Literature | |
| 6. | ALA4005618 | B | Inhibition of PRDM9 (unknown origin) at 10 uM using biotin-labeled peptide as substrate and [3H]-SAM measured after 1 hr by scintillation proximity assay | Homo sapiens | 1 | ALA4004823 | single protein format | Scientific Literature | |
| 7. | ALA4005647 | B | Inhibition of PRDM9 (unknown origin) at 1 uM using biotin-labeled peptide as substrate and [3H]-SAM measured after 1 hr by scintillation proximity assay | Homo sapiens | 1 | ALA4004823 | single protein format | Scientific Literature | |
| 8. | ALA4026511 | B | Inhibition of PRDM9 (unknown origin) at 50 uM incubated for 15 mins followed by substrate addition measured after 60 mins by AlphaLisa method | Homo sapiens | 1 | ALA4024748 | single protein format | Scientific Literature | |
| 9. | ALA4026519 | B | Inhibition of PRDM9 (unknown origin) at 100 uM incubated for 15 mins followed by substrate addition measured after 60 mins by AlphaLisa method | Homo sapiens | 1 | ALA4024748 | single protein format | Scientific Literature | |
| 10. | ALA4346623 | B | Inhibition of PRDM9 (unknown origin) assessed as reduction in incorporation of [3H]-labeled methyl group into biotinylated substrate using [3H-SAM] at 10 uM incubated for 1 hr by scintillation proximity assay | Homo sapiens | 1 | ALA4342528 | single protein format | Scientific Literature | |
| 11. | ALA4377304 | B | Inhibition of human PRDM9 up to 50 uM using Biot-H3 (1-25) as substrate and in presence of [3H]-SAM incubated for 1 hr by scintillation proximity assay | Homo sapiens | 1 | ALA4376809 | single protein format | Scientific Literature | |
| 12. | ALA4480231 | B | Inhibition of PRDM9 (unknown origin) using biotin-labeled histone substrate assessed as residual activity at 50 uM in presence of [3H-Me]SAM by scintillation proximity assay relative to control | Homo sapiens | 24 | ALA4477270 | single protein format | Scientific Literature | |
| 13. | ALA4731565 | B | Inhibition of recombinant human N-terminal GST-tagged PRDM9 (2 to 414 residues) expressed in baculovirus infected Sf9 cells using histone H3 as substrate at 10 uM by radiometric HotSpot assay relative to control | Homo sapiens | 1 | ALA4725473 | cell-based format | Scientific Literature | |
| 14. | ALA5030807 | B | Inhibition of PRDM9 (unknown origin) at 1 to 10 uM | Homo sapiens | 2 | ALA5030506 | single protein format | Scientific Literature | |
| 15. | ALA5119843 | B | Inhibition of human recombinant PRDM9 (2 to 414 residues) expressed in Sf9 insect cells at 10 uM using histone as substrate by scintillation/filter assay | Homo sapiens | 1 | ALA5113528 | cell-based format | Scientific Literature | |
| 16. | ALA5119880 | B | Inhibition of human recombinant PRDM9 (2 to 414 residues) expressed in Sf9 insect cells at 50 uM using histone as substrate by scintillation/filter assay relative to control | Homo sapiens | 1 | ALA5113528 | cell-based format | Scientific Literature | |
| 17. | ALA5210291 | B | Affinity On-target Cellular interaction (Western Blot (inhibition of PRDM9-dependent trimethylation of ectopic H3K4 in HEK293T cells)) EUB0000234b PRDM9 | Homo sapiens | 1 | ALA5210121 | cell-based format | Literature data from EUbOPEN Chemogenomic Library | |
| 18. | ALA5210597 | B | Affinity Biochemical interaction (Scintillation proximity assay (SPA)) EUB0000234b PRDM9 | Homo sapiens | 1 | ALA5210307 | single protein format | Literature data from EUbOPEN Chemogenomic Library | |
| 19. | ALA5214657 | B | Selectivity interaction (Methyltransferase panel (DSF assay)) EUB0000234b PRDM9 | Homo sapiens | 1 | ALA5212743 | single protein format | Literature data from EUbOPEN Chemogenomic Library | |
| 20. | ALA5214658 | B | Selectivity interaction (NanoLuciferase thermal shift assay (NALTSA, in HEK293 cells)) EUB0000234b PRDM9 | Homo sapiens | 1 | ALA5212743 | cell-based format | Literature data from EUbOPEN Chemogenomic Library |
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