| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3592411 | B | Inhibition of NSD1 (unknown origin) at 1 uM after 1 hr by filter-based assay | Homo sapiens | 1 | ALA3588844 | single protein format | Scientific Literature | |
| 2. | ALA3626820 | B | Inhibition of NSD1 (unknown origin) at 100 uM preincubated for 15 mins followed by substrate/[3H]-SAM addition measured after 4 hrs by liquid scintillation counting analysis relative to control | Homo sapiens | 2 | ALA3621043 | single protein format | Scientific Literature | |
| 3. | ALA3784089 | B | Inhibition of human NSD1 at 10 and 50 uM | Homo sapiens | 1 | ALA3779843 | single protein format | Scientific Literature | |
| 4. | ALA3803126 | B | Inhibition of NSD1 (unknown origin) at 10 uM relative to control | Homo sapiens | 2 | ALA3797202 | single protein format | Scientific Literature | |
| 5. | ALA3821914 | B | Inhibition of NSD1 (unknown origin) at 1 to 50 uM by TCA precipitation assay | Homo sapiens | 1 | ALA3817823 | single protein format | Scientific Literature | |
| 6. | ALA3859062 | B | Inhibition of NSD1 (unknown origin) at 50 uM using biotin-labeled peptide as substrate and [3H]-SAM measured after 1 hr by scintillation proximity assay | Homo sapiens | 1 | ALA3856251 | single protein format | Scientific Literature | |
| 7. | ALA4006082 | B | Inhibition of NSD1 (unknown origin) at 50 and 100 uM preincubated for 15 mins followed by substrate and [3H]-SAM addition after 120 mins by MicroBeta counting | Homo sapiens | 1 | ALA4004835 | single protein format | Scientific Literature | |
| 8. | ALA4013554 | B | Inhibition of NSD1 (unknown origin) preincubated for 15 mins followed by [3H]-SAM addition measured after 4 hrs by liquid scintillation counting | Homo sapiens | 1 | ALA4011642 | single protein format | Scientific Literature | |
| 9. | ALA4346638 | B | Inhibition of NSD1 (unknown origin) at 10 uM using [3H-SAM] and nucleosome as substrate incubated for 1 hr by scintillation proximity assay | Homo sapiens | 1 | ALA4342528 | single protein format | Scientific Literature | |
| 10. | ALA4377327 | B | Inhibition of human NSD1 up to 50 uM using chicken nucleosome as substrate and in presence of [3H]-SAM incubated for 1 hr by filter-based assay | Homo sapiens | 1 | ALA4376809 | single protein format | Scientific Literature | |
| 11. | ALA4480238 | B | Inhibition of NSD1 (unknown origin) using biotin-labeled histone substrate assessed as residual activity at 50 uM in presence of [3H-Me]SAM by scintillation proximity assay relative to control | Homo sapiens | 24 | ALA4477270 | single protein format | Scientific Literature | |
| 12. | ALA4628787 | B | Inhibition of NSD1 (unknown origin) at 100 uM | Homo sapiens | 1 | ALA4627335 | single protein format | Scientific Literature | |
| 13. | ALA4731586 | B | Inhibition of N-terminal His-tagged recombinant human NSD1 (1538 to 2696 residues) expressed in baculovirus infected insect cells using nucleosome as substrate at expressed in 10 uM by radiometric HotSpot assay relative to control | Homo sapiens | 1 | ALA4725473 | cell-based format | Scientific Literature | |
| 14. | ALA4827173 | B | Inhibition of NSD1 (unknown origin) using SAM as substrate preincubated for 10 mins followed by substrate addition measured after 4 hrs by AlphaLISA method | Homo sapiens | 1 | ALA4825702 | single protein format | Scientific Literature | |
| 15. | ALA4827267 | B | Inhibition of human NSD1-SET using histone H3.1 as substrate incubated for 1 hr by Western blot analysis | Homo sapiens | 1 | ALA4825702 | single protein format | Scientific Literature | |
| 16. | ALA4833661 | B | Inhibition of NSD1 (unknown origin) at 10 uM using SAM as substrate measured up to 960 mins by AlphaScreen microplate reader assay relative to control | Homo sapiens | 1 | ALA4831544 | single protein format | Scientific Literature | |
| 17. | ALA5030818 | B | Inhibition of NSD1 (unknown origin) at 1 to 10 uM | Homo sapiens | 2 | ALA5030506 | single protein format | Scientific Literature | |
| 18. | ALA5119840 | B | Inhibition of human recombinant N-terminal his-tagged NSD1 (1538 to 2696 residues) expressed in Sf9 insect cells at 10 uM by scintillation/filter assay | Homo sapiens | 1 | ALA5113528 | cell-based format | Scientific Literature | |
| 19. | ALA5119877 | B | Inhibition of human recombinant N-terminal his-tagged NSD1 (1538 to 2696 residues) expressed in Sf9 insect cells at 50 uM by scintillation/filter assay relative to control | Homo sapiens | 1 | ALA5113528 | cell-based format | Scientific Literature | |
| 20. | ALA5129694 | B | Inhibition of N-terminal His-tagged NSD1 (1538 to 2696 residues) (unknown origin) expressed in baculovirus expression system at 1 uM using 3H-SAM as a substrate relative to control | Homo sapiens | 1 | ALA5126600 | assay format | Scientific Literature |
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