| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3632282 | B | Inhibition of CAMK1beta (unknown origin) at 10 uM after 120 mins P33 radiolabeled kinase activity assay | Homo sapiens | 3 | ALA3627608 | single protein format | Scientific Literature | |
| 2. | ALA3748642 | B | Inhibition of human CAMK1beta using [KKALRRQETVDAL] as substrate | Homo sapiens | 1 | ALA3745707 | single protein format | Scientific Literature | |
| 3. | ALA3817220 | B | Inhibition of human CAMK1beta at 1 uM using [KKALRRQETVDAL] as substrate | Homo sapiens | 1 | ALA3813650 | single protein format | Scientific Literature | |
| 4. | ALA4025036 | B | Inhibition of wild-type human partial length CAMK1B (W9 to A311 residues) expressed in mammalian expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4024706 | assay format | Scientific Literature | |
| 5. | ALA4043847 | B | Inhibition of wild-type human partial length CAMK1B (W9 to A311 residues) expressed in HEK293 cells assessed as residual activity at 1000 nM after 30 mins by Kinomescan method relative to control | Homo sapiens | 1 | ALA4043093 | cell-based format | Scientific Literature | |
| 6. | ALA4156926 | B | Binding affinity to wild-type human partial length CAMK1B (W9 to A311 residues) expressed in mammalian expression system assessed as residual binding at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4152344 | assay format | Scientific Literature | |
| 7. | ALA4185705 | B | Binding affinity to wild-type human partial length CAMK1B (W9 to A311 residues) expressed in HEK293 cells at 1 uM by Kinomescan method relative to control | Homo sapiens | 2 | ALA4184148 | cell-based format | Scientific Literature | |
| 8. | ALA4190894 | B | Inhibition of recombinant full-length human CAMK1beta at 1 uM using KKLRRTLSFAEPG as substrate after 40 mins in presence of [gamma-33P]ATP by scintillation counting method | Homo sapiens | 1 | ALA4190187 | single protein format | Scientific Literature | |
| 9. | ALA4230605 | B | Binding affinity to wild-type human partial length CAMK1B (W9 to A311 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4229344 | assay format | Scientific Literature | |
| 10. | ALA4264194 | B | Binding affinity to wild-type human partial length CAMK1B (W9 to A311 residues) expressed in mammalian expression system assessed as remaining unbound target protein level at 1000 nM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4261600 | assay format | Scientific Literature | |
| 11. | ALA4314615 | B | Inhibition of recombinant full-length human CaMK1beta assessed as residual activity at 10 uM using calmodulin as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation counting method | Homo sapiens | 1 | ALA4311992 | single protein format | Scientific Literature | |
| 12. | ALA4327605 | B | Inhibition of human CAMK1B assessed as residual activity at 1 uM using KKALRRQETVDAL as substrate by [gamma-33P]-ATP assay relative to control | Homo sapiens | 2 | ALA4325871 | single protein format | Scientific Literature | |
| 13. | ALA4327966 | B | Inhibition of human CAMK1B assessed as residual activity at 100 uM using KKALRRQETVDAL as substrate by [gamma-33P]-ATP assay relative to control | Homo sapiens | 1 | ALA4325871 | single protein format | Scientific Literature | |
| 14. | ALA4328330 | B | Inhibition of human CAMK1B using KKALRRQETVDAL as substrate by [gamma-33P]-ATP assay | Homo sapiens | 1 | ALA4325871 | single protein format | Scientific Literature | |
| 15. | ALA4334987 | B | Inhibition of recombinant full length human CaMKIbeta assessed as residual activity at 1 uM using KKLRRTLSFAEP as substrate incubated for 40 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay relative to control | Homo sapiens | 2 | ALA4334438 | single protein format | Scientific Literature | |
| 16. | ALA4336815 | B | Inhibition of recombinant full length human CaMKIbeta assessed as residual activity at 10 uM using KKLRRTLSFAEP as substrate incubated for 40 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay relative to control | Homo sapiens | 1 | ALA4334471 | single protein format | Scientific Literature | |
| 17. | ALA4351767 | B | Inhibition of recombinant full-length human CaMK1beta at 10 uM using calmodulin as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation counting method | Homo sapiens | 1 | ALA4350961 | single protein format | Scientific Literature | |
| 18. | ALA4352292 | B | Inhibition of human CAMK1B at 10 uM using KKALRRQETVDAL as substrate in presence of [gamma-33P]-ATP | Homo sapiens | 1 | ALA4350963 | single protein format | Scientific Literature | |
| 19. | ALA4357783 | B | Binding affinity to wild-type human partial length CAMK1B (W9 to A311 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4354843 | assay format | Scientific Literature | |
| 20. | ALA4366308 | B | Inhibition of human CAMK1B at 100 nM using KKALRRQETVDAL as substrate by [gamma-33P]-ATP assay | Homo sapiens | 1 | ALA4364276 | single protein format | Scientific Literature |
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