# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3734501 | Binding | Inhibition of recombinant human PKG1alpha using fluorescein-labeled peptide as substrate by fluorescence-electrophoretic mobility shift assay | Homo sapiens | 1 | ALA3727354 | single protein format | Patent Bioactivity Data | |
2. | ALA3750013 | Binding | Inhibition of human PKG1alpha using [LRRASLG] as substrate | Homo sapiens | 1 | ALA3745707 | single protein format | Scientific Literature | |
3. | ALA3750014 | Binding | Inhibition of human PKG1beta using [LRRASLG] as substrate | Homo sapiens | 1 | ALA3745707 | single protein format | Scientific Literature | |
4. | ALA3750458 | Binding | Inhibition of PKG1alpha (unknown origin) at 1 uM | Homo sapiens | 1 | ALA3745631 | single protein format | Scientific Literature | |
5. | ALA3761164 | Binding | Inhibition of PKG1alpha (unknown origin) at 100 nM | Homo sapiens | 1 | ALA3758169 | single protein format | Scientific Literature | |
6. | ALA3777522 | Binding | Inhibition of N-terminal His6-tagged recombinant human PKG1alpha expressed in baculovirus infected insect Sf9 cells assessed as remaining activity at 1 uM relative to control | Homo sapiens | 3 | ALA3774357 | cell-based format | Scientific Literature | |
7. | ALA3777523 | Binding | Inhibition of N-terminal His6-tagged recombinant human PKG1beta expressed in baculovirus infected insect Sf9 cells assessed as remaining activity at 1 uM relative to control | Homo sapiens | 3 | ALA3774357 | cell-based format | Scientific Literature | |
8. | ALA3802468 | Binding | Inhibition of partial length wild type human PRKG1 expressed in bacterial system assessed as enzyme activity at 1 uM relative to control | Homo sapiens | 1 | ALA3797029 | assay format | Scientific Literature | |
9. | ALA3807488 | Binding | Inhibition of PRKG1 (unknown origin) at 10 uM by mobility shift assay | Homo sapiens | 1 | ALA3804794 | single protein format | Scientific Literature | |
10. | ALA3807605 | Binding | Inhibition of PRKG1 (unknown origin) at 0.5 uM by mobility shift assay | Homo sapiens | 1 | ALA3804794 | single protein format | Scientific Literature | |
11. | ALA3807899 | Binding | Inhibition of PRKG1 (unknown origin) by mobility shift assay | Homo sapiens | 1 | ALA3804794 | single protein format | Scientific Literature | |
12. | ALA3815960 | Binding | Inhibition of human PKG1alpha at 1 uM using [LRRASLG] as substrate | Homo sapiens | 1 | ALA3813650 | single protein format | Scientific Literature | |
13. | ALA3815961 | Binding | Inhibition of human PKG1beta at 1 uM using [LRRASLG] as substrate | Homo sapiens | 1 | ALA3813650 | single protein format | Scientific Literature | |
14. | ALA3816507 | Binding | Inhibition of full length recombinant human GST-tagged PKG1alpha expressed in baculovirus expression system at 1 uM relative to control | Homo sapiens | 1 | ALA3813614 | assay format | Scientific Literature | |
15. | ALA1071351 | Binding | Residual activity of PRKG1 at 10 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
16. | ALA1065746 | Binding | Inhibition of PRKG1 | 2 | ALA1157712 | single protein format | Scientific Literature | ||
17. | ALA1101492 | Binding | Inhibition of PRKG1 at 10 uM | 2 | ALA1154277 | single protein format | Scientific Literature | ||
18. | ALA1166828 | Binding | Inhibition of PRKG1 at 1 uM | 10 | ALA1165965 | single protein format | Scientific Literature | ||
19. | ALA1175238 | Binding | Inhibition of PRKG1 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
20. | ALA1176572 | Binding | Inhibition of PKG1alpha at 1 uM | 1 | ALA1177702 | single protein format | Scientific Literature |