# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3777493 | Binding | Inhibition of N-terminal GST-tagged mouse MKK4 expressed in Escherichia coli assessed as remaining activity at 1 uM relative to control | Mus musculus | 3 | ALA3774357 | assay format | Scientific Literature | |
2. | ALA854390 | Binding | Residual activity at mouse MKK4 at 10 uM in presence of 10 uM ATP relative to control | Mus musculus | 1 | ALA1138050 | single protein format | Scientific Literature | |
3. | ALA854693 | Binding | Percentage activity of mouse MKK4 in the presence of 10 uM of compound and 10 uM of ATP in comparison with control | Mus musculus | 1 | ALA1137942 | single protein format | Scientific Literature | |
4. | ALA886989 | Binding | Inhibition of mouse MKK4 Met at 1 uM relative to control | Mus musculus | 4 | ALA1139192 | single protein format | Scientific Literature | |
5. | ALA1249694 | Binding | Inhibition of mouse MKK4 activity at 10 uM by radiometric assay | Mus musculus | 2 | ALA1240306 | single protein format | Scientific Literature | |
6. | ALA921995 | Binding | Activity of mouse MKK4 kinase at 1 uM | Mus musculus | 1 | ALA1147076 | single protein format | Scientific Literature | |
7. | ALA732666 | Binding | Inhibition of Mitogen activated protein kinase kinase 4 | Mus musculus | 3 | ALA1146654 | single protein format | Scientific Literature | |
8. | ALA732810 | Binding | Inhibition of mouse Mitogen activated protein kinase kinase 4 at 10 uM | Mus musculus | 2 | ALA1145082 | single protein format | Scientific Literature | |
9. | ALA1646197 | Binding | Inhibition of mouse MKK4 at 10 uM after 60 mins by TR-FRET assay | Mus musculus | 1 | ALA1641539 | single protein format | Scientific Literature | |
10. | ALA2166395 | Binding | Inhibition of mouse MKK4 at 10 uM | Mus musculus | 1 | ALA2163300 | single protein format | Scientific Literature | |
11. | ALA3101405 | Binding | Inhibition of mouse MKK4 assessed as residual activity at 1 uM relative to control | Mus musculus | 1 | ALA3098105 | single protein format | Scientific Literature | |
12. | ALA3242552 | Binding | Inhibition of mouse MKK4 assessed as enzyme activity at 1 uM relative to control | Mus musculus | 1 | ALA3232845 | single protein format | Scientific Literature | |
13. | ALA3292191 | Binding | Inhibition of mouse MKK4 assessed as residual activity at 10 uM relative to control | Mus musculus | 2 | ALA3286226 | single protein format | Scientific Literature | |
14. | ALA4191060 | Binding | Inhibition of recombinant mouse MKK4 (34 to end residues) at 1 uM using inactive JNK1a1 as substrate after 40 mins in presence of [gamma-33P]ATP by scintillation counting method | Mus musculus | 1 | ALA4190187 | single protein format | Scientific Literature | |
15. | ALA4337195 | Binding | Inhibition of recombinant mouse MKK4 (34 to end residues) assessed as residual activity at 10 uM using poly(Glu, Tyr) 4:1 as substrate incubated for 40 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay relative to control | Mus musculus | 1 | ALA4334471 | single protein format | Scientific Literature | |
16. | ALA4408044 | Binding | Inhibition of recombinant mouse MKK4 (34 to end residues) at 1 uM using unactive JNK1a1 as substrate incubated for 40 mins in presence of [gamma-33P]-ATP by scintillation counting method relative to control | Mus musculus | 1 | ALA4406821 | single protein format | Scientific Literature | |
17. | ALA4814583 | Binding | Binding affinity to GST tagged mouse MKK4 expressed in Escherichia coli expression system assessed as residual activity at 100 nM measured by Kinomescan assay | Mus musculus | 67 | ALA4813918 | assay format | Scientific Literature | |
18. | ALA4814587 | Binding | Binding affinity to GST tagged mouse MKK4 expressed in Escherichia coli expression system measured by Kinomescan assay | Mus musculus | 4 | ALA4813918 | assay format | Scientific Literature | |
19. | ALA4880678 | Binding | MKK4 (m) Millipore kinase activity assay | Homo sapiens | 1 | ALA4507263 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
20. | ALA4881541 | Binding | MKK4 (m) Upstate kinase activity assay | Mus musculus | 1 | ALA4507274 | single protein format | Donated Chemical Probes - SGC Frankfurt |