# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA680869 | B | Inhibition of the (-40 mV) current elicited by 100 uM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | 20 | cell-based format | Scientific Literature | |||
2. | ALA680870 | B | Inhibition of the (-80 mV) current elicited by 100 uM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | 20 | cell-based format | Scientific Literature | |||
3. | ALA884410 | B | Electrophysiological data on Xenopus oocytes, expressing homomeric Ionotropic glutamate receptor AMPA 1 (GluR1o) | Xenopus laevis | 3 | cell-based format | Scientific Literature | ||
4. | ALA701238 | B | In vitro inhibitory activity against Ionotropic glutamate receptor AMPA 1 of HEK293 cells in FLIPR assay | 2 | cell-based format | Scientific Literature | |||
5. | ALA701239 | B | Ability to displace binding of [3H]AMPA to recombinant human Ionotropic glutamate receptor AMPA 1 | 3 | single protein format | Scientific Literature | |||
6. | ALA878883 | B | Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 1 expressed in HEK293 cells | Homo sapiens | 14 | cell-based format | Scientific Literature | ||
7. | ALA701240 | B | Binding affinity of compound was determined against Ionotropic glutamate receptor AMPA 1 using cell membranes prepared from HEK293 cells | 7 | cell-based format | Scientific Literature | |||
8. | ALA701241 | B | Compound was tested for binding affinity against human Ionotropic glutamate receptor AMPA 1 in HEK293 cells using [3H]-AMPA as radioligand | 4 | cell-based format | Scientific Literature | |||
9. | ALA701247 | B | Binding affinity of compound was determined towards cloned Ionotropic glutamate receptor AMPA 1 (GluR1) expressed in Sf 9 insect cells | 3 | cell-based format | Scientific Literature | |||
10. | ALA829619 | B | Binding affinity for ionotropic Glutamate receptor AMPA 1 expressed in Sf9 cells | 5 | cell-based format | Scientific Literature | |||
11. | ALA863279 | F | Inhibitory effect on glutamate-induced calcium influx at homomeric human GLUA1 receptor expressed in HEK293 cells up to 300 uM | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
12. | ALA865008 | F | Inhibition of glutamate-induced calcium influx in HEK293 cells expressing human GLUA1 up to 100 uM | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
13. | ALA865014 | F | Inhibition of glutamate-induced calcium influx in HEK293 cells expressing human GLUA1 | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
14. | ALA934442 | B | Binding affinity at iGluR1o receptor expressed in sf9 cells by radioligand binding assay | 2 | cell-based format | Scientific Literature | |||
15. | ALA895662 | F | Agonist activity at GluR1 expressed in HEK293 cells by Fluo-4/Ca2+ assay | 6 | cell-based format | Scientific Literature | |||
16. | ALA895663 | F | Agonist activity at GluR1 expressed in HEK293 cells relative to S-Glutamate by Fluo-4/Ca2+ assay | 4 | cell-based format | Scientific Literature | |||
17. | ALA895670 | F | Agonist activity at GluR1 D399S mutant expressed in HEK293 cells by Fluo-4/Ca2+ assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
18. | ALA895671 | F | Agonist activity at GluR1 D399S mutant expressed in HEK293 cells up to 3 mM by Fluo-4/Ca2+ assay relative to S-Glutamate | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
19. | ALA895672 | F | Agonist activity at GluR1 E683A mutant expressed in HEK293 cells by Fluo-4/Ca2+ assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
20. | ALA895673 | F | Agonist activity at GluR1 E683A mutant expressed in HEK293 cells up to 3 mM by Fluo-4/Ca2+ assay relative to S-Glutamate | Homo sapiens | 1 | cell-based format | Scientific Literature |