# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA679557 | B | Inhibitory activity against human sodium and chloride dependent GABA transporter 3 | 25 | ALA1127589 | single protein format | Scientific Literature | ||
2. | ALA679558 | B | Compound was evaluated for inhibitory activity against human Sodium- and chloride-dependent GABA transporter 3 | 3 | ALA1127589 | single protein format | Scientific Literature | ||
3. | ALA677769 | F | Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human GAT-3 transporter | 5 | ALA1129108 | assay format | Scientific Literature | ||
4. | ALA1166721 | B | Binding affinity to GAT3 | 4 | ALA1165889 | single protein format | Scientific Literature | ||
5. | ALA1647452 | B | Inhibition of GAT3 | 1 | ALA1641586 | single protein format | Scientific Literature | ||
6. | ALA1663481 | B | Inhibition of [3H]GABA uptake at GAT3 expressed in HEK cells | 18 | ALA1649378 | cell-based format | Scientific Literature | ||
7. | ALA1663482 | B | Inhibition of [3H]GABA uptake at GAT3 expressed in HEK cells at 100 uM | 5 | ALA1649378 | cell-based format | Scientific Literature | ||
8. | ALA1776008 | B | Inhibition of human GAT3-mediated GABA uptake | Homo sapiens | 1 | ALA1773002 | single protein format | Scientific Literature | |
9. | ALA1918361 | B | Inhibition of human GAT3 assessed as [3H]GABA uptake | Homo sapiens | 1 | ALA1914421 | single protein format | Scientific Literature | |
10. | ALA2208547 | B | Inhibition of human GAT3 expressed in tcA201 cells assessed as inhibition of [3H]GABA uptake at 1 mM after 3 mins by scintillation counting | Homo sapiens | 1 | ALA2203122 | cell-based format | Scientific Literature | |
11. | ALA2417028 | B | Inhibition of human GAT3 transfected in CHO cells assessed as [3H]GABA uptake after 20 mins by liquid scintillation counting analysis | Homo sapiens | 5 | ALA2413054 | cell-based format | Scientific Literature | |
12. | ALA2417032 | B | Inhibition of human GAT3 transfected in CHO cells assessed as [3H]GABA uptake at 100 uM after 20 mins by liquid scintillation counting analysis | Homo sapiens | 8 | ALA2413054 | cell-based format | Scientific Literature | |
13. | ALA2433116 | B | Inhibition of GAT-3 (unknown origin) expressed in african green monkey COS7 cells using [3H]-GABA as substrate after 10 mins by scintillation counting | Homo sapiens | 1 | ALA2429840 | cell-based format | Scientific Literature | |
14. | ALA3363498 | B | Inhibition of human GAT3 transfected in CHO cells assessed as [3H]GABA uptake after 20 mins by liquid scintillation counting analysis | Homo sapiens | 5 | ALA3351485 | cell-based format | Scientific Literature | |
15. | ALA3363504 | B | Inhibition of human GAT3 transfected in CHO cells assessed as [3H]GABA uptake at 100 uM after 20 mins by liquid scintillation counting analysis | Homo sapiens | 3 | ALA3351485 | cell-based format | Scientific Literature | |
16. | ALA3877716 | B | Inhibition of human GAT-3 expressed in thymidine kinase deficient mouse LM cells assessed as decrease in [3H]GABA uptake after 10 mins by scintillation counter method | Homo sapiens | 1 | ALA3877251 | cell-based format | Scientific Literature | |
17. | ALA4031690 | B | Inhibition of human GAT3 L314Q mutant expresses in tsA201 cells assessed as reduction in [3H]GABA uptake after 3 mins by scintillation counting method | Homo sapiens | 3 | ALA4028872 | cell-based format | Scientific Literature | |
18. | ALA4031699 | B | Inhibition of human GAT3 expresses in tsA201 cells assessed as reduction in [3H]GABA uptake after 3 mins by scintillation counting method | Homo sapiens | 32 | ALA4028872 | cell-based format | Scientific Literature | |
19. | ALA4031735 | B | Inhibition of human GAT3 S468Y mutant expresses in tsA201 cells assessed as reduction in [3H]GABA uptake after 3 mins by scintillation counting method | Homo sapiens | 3 | ALA4028872 | cell-based format | Scientific Literature | |
20. | ALA4267186 | B | Inhibition of human GAT3 expressed in CHO cells assessed as reduction in [3H]GABA uptake at 100 uM after 20 mins by liquid scintillation counting analysis relative to control | Homo sapiens | 8 | ALA4265902 | cell-based format | Scientific Literature |