# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA817081 | B | In vitro inhibition of [3H]AVP binding to human V2 receptor from murine fibroblast cell line (LV2) | 5 | ALA1131757 | cell-based format | Scientific Literature | ||
2. | ALA817082 | B | Inhibition constant for vasopressin-stimulated adenylate cyclase of medullary membranes of human kidney | 6 | ALA1124391 | assay format | Scientific Literature | ||
3. | ALA817083 | B | Inhibition constant for vasopressin-stimulated adenylate cyclase of medullary membranes of human kidney; NT=Not tested | 3 | ALA1124391 | assay format | Scientific Literature | ||
4. | ALA818586 | F | Inhibition of 1 nM AVP-induced cAMP accumulation in cells expressing human vasopressin V2 receptor | 22 | ALA1146755 | assay format | Scientific Literature | ||
5. | ALA818587 | B | Inhibition of [3H]AVP binding to recombinant human vasopressin V2 receptor | 32 | ALA1146755 | single protein format | Scientific Literature | ||
6. | ALA873234 | F | In vitro antagonist activity was measured by inhibition of vasopressin-stimulated adenylate cyclase in renal medullary preparation in dog | Canis lupus familiaris | 4 | ALA1124168 | tissue-based format | Scientific Literature | |
7. | ALA817655 | F | Percentage of maximal cAMP accumulation at a concentration of 10e-4 M was done in HeLa cells expressing the human Vasopressin V2 receptor | 1 | ALA1135753 | cell-based format | Scientific Literature | ||
8. | ALA816919 | F | Percentage of maximal cAMP accumulation at a concentration of 10e-6 M was done in HeLa cells expressing the human Vasopressin V2 receptor | 2 | ALA1135753 | cell-based format | Scientific Literature | ||
9. | ALA816920 | B | Ability to displace [3H]arginine vasopressin in cloned human V2 receptor | Homo sapiens | 10 | ALA1136360 | single protein format | Scientific Literature | |
10. | ALA817831 | B | Ability to displace [3H]arginine vasopressin in cloned human V2 receptor at 0.2 uM | Homo sapiens | 1 | ALA1136360 | single protein format | Scientific Literature | |
11. | ALA817832 | B | Binding affinity measured by inhibition of 3[H] AVP binding to cloned human V2 receptor (Compound 7o) | 1 | ALA1146639 | single protein format | Scientific Literature | ||
12. | ALA817833 | B | Binding affinity measured by inhibition of 3[H] AVP binding to cloned human vasopressin V2 receptor | 16 | ALA1146639 | single protein format | Scientific Literature | ||
13. | ALA817834 | B | Binding affinity against human Vasopressin V2 receptor expressed in HeLa cells was determined | 3 | ALA1135753 | cell-based format | Scientific Literature | ||
14. | ALA817835 | F | Inhibition of vasopressin induced cAMP accumulation in human V2 receptor expressing cells | Homo sapiens | 6 | ALA1136360 | assay format | Scientific Literature | |
15. | ALA817836 | F | Inhibition of vasopressin induced cAMP accumulation in human V2 receptor expressing cells; ND= Not determined | Homo sapiens | 5 | ALA1136360 | assay format | Scientific Literature | |
16. | ALA817837 | B | Displacement of [3H]AVP from human V2 receptors expressed in HEK293 cells | Homo sapiens | 13 | ALA1136603 | cell-based format | Scientific Literature | |
17. | ALA817838 | B | In vitro binding affinity to human V2 receptor | Homo sapiens | 10 | ALA1133322 | single protein format | Scientific Literature | |
18. | ALA817839 | B | In vitro binding affinity to human V2 receptor; not tested | Homo sapiens | 8 | ALA1133322 | single protein format | Scientific Literature | |
19. | ALA817840 | B | Displacement of [3H]AVP from human vasopressin V2-receptor expressed in murine fibroblast cell (LV2) membranes | Homo sapiens | 13 | ALA1133037 | cell-based format | Scientific Literature | |
20. | ALA873374 | B | Compound was tested in vitro for its ability to displace 3H AVP in membrane preparation from murine fibroblast cell line (LV2) expressing the human vasopressin V2-receptor; Not tested | 1 | ALA1133037 | cell-based format | Scientific Literature |