# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA696972 | B | In vitro inhibitory activity against Ionotropic glutamate receptor AMPA 2 of HEK293 cells in FLIPR assay | 2 | cell-based format | Scientific Literature | |||
2. | ALA696973 | B | Ability to displace binding of [3H]AMPA to recombinant human Ionotropic glutamate receptor AMPA 2 | 3 | single protein format | Scientific Literature | |||
3. | ALA696974 | B | Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 2 expressed in HEK293 cells | Homo sapiens | 14 | cell-based format | Scientific Literature | ||
4. | ALA696975 | B | Binding affinity of compound was determined against Ionotropic glutamate receptor AMPA 2 using cell membranes prepared from HEK293 cells | 7 | cell-based format | Scientific Literature | |||
5. | ALA696976 | B | Compound was tested for binding affinity against human Ionotropic glutamate receptor AMPA 2 in HK293 cells using [3H]AMPA as radioligand | 4 | cell-based format | Scientific Literature | |||
6. | ALA697507 | B | Binding affinity of compound was determined towards cloned Ionotropic glutamate receptor AMPA 2 (GluR2) expressed in Sf 9 insect cells | 3 | cell-based format | Scientific Literature | |||
7. | ALA829620 | B | Binding affinity for ionotropic Glutamate receptor AMPA 2 expressed in Sf9 cells | 5 | cell-based format | Scientific Literature | |||
8. | ALA840052 | B | Inhibition of [3H]AMPA binding to human Ionotropic glutamate receptor 2 | Homo sapiens | 1 | single protein format | Scientific Literature | ||
9. | ALA829051 | B | Inhibition of [3H]-AMPA binding to human GluR2 receptors expressed in HEK 293 cells | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
10. | ALA863280 | F | Inhibitory effect on glutamate-induced calcium influx at homomeric human GLUA2 receptor expressed in HEK293 cells up to 300 uM | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
11. | ALA865009 | F | Inhibition of glutamate-induced calcium influx in HEK293 cells expressing human GLUA2 up to 100 uM | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
12. | ALA865015 | F | Inhibition of glutamate-induced calcium influx in HEK293 cells expressing human GLUA2 | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
13. | ALA871564 | F | Activity against human GLUR2 flip expressed in HEK293 cells assessed as glutamate-stimulated calcium influx by FLIPR assay | Homo sapiens | 20 | cell-based format | Scientific Literature | ||
14. | ALA871565 | F | Activity against human GLUR2 flop expressed in HEK293 cells assessed as glutamate-stimulated calcium influx by FLIPR assay | Homo sapiens | 20 | cell-based format | Scientific Literature | ||
15. | ALA856920 | F | Activity at human recombinant iGluR2 flip expressed in HEK293 cells measured as change in intracellular calcium ion concentration in presence of glutamate by FLIPR assay | Homo sapiens | 25 | cell-based format | Scientific Literature | ||
16. | ALA856924 | F | Activity at human recombinant iGluR2 flop expressed in HEK293 cells measured as change in intracellular calcium ion concentration in presence of glutamate by FLIPR assay | Homo sapiens | 25 | cell-based format | Scientific Literature | ||
17. | ALA914410 | F | Antagonist activity at human recombinant GLUA2-AMPA receptor expressed in HEK293 cells assessed as inhibition of glutamate-stimulated calcium influx by FLIPR assay | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
18. | ALA895664 | F | Agonist activity at GluR2Q expressed in HEK293 cells by Fluo-4/Ca2+ assay | 6 | cell-based format | Scientific Literature | |||
19. | ALA895665 | F | Agonist activity at GluR2Q expressed in HEK293 cells relative to S-Glutamate by Fluo-4/Ca2+ assay | 4 | cell-based format | Scientific Literature | |||
20. | ALA934441 | B | Binding affinity at iGluR2 receptor S1S2J domain expressed in sf9 cells by radioligand binding assay | 2 | cell-based format | Scientific Literature |