# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA696972 | B | In vitro inhibitory activity against Ionotropic glutamate receptor AMPA 2 of HEK293 cells in FLIPR assay | 2 | ALA1145950 | cell-based format | Scientific Literature | ||
2. | ALA696973 | B | Ability to displace binding of [3H]AMPA to recombinant human Ionotropic glutamate receptor AMPA 2 | 3 | ALA1136004 | single protein format | Scientific Literature | ||
3. | ALA696974 | B | Displacement of [3H]AMPA from human Ionotropic glutamate receptor AMPA 2 expressed in HEK293 cells | Homo sapiens | 14 | ALA1130220 | cell-based format | Scientific Literature | |
4. | ALA696975 | B | Binding affinity of compound was determined against Ionotropic glutamate receptor AMPA 2 using cell membranes prepared from HEK293 cells | 7 | ALA1133269 | cell-based format | Scientific Literature | ||
5. | ALA696976 | B | Compound was tested for binding affinity against human Ionotropic glutamate receptor AMPA 2 in HK293 cells using [3H]AMPA as radioligand | 4 | ALA1133179 | cell-based format | Scientific Literature | ||
6. | ALA697507 | B | Binding affinity of compound was determined towards cloned Ionotropic glutamate receptor AMPA 2 (GluR2) expressed in Sf 9 insect cells | 3 | ALA1144891 | cell-based format | Scientific Literature | ||
7. | ALA829620 | B | Binding affinity for ionotropic Glutamate receptor AMPA 2 expressed in Sf9 cells | 5 | ALA1144430 | cell-based format | Scientific Literature | ||
8. | ALA840052 | B | Inhibition of [3H]AMPA binding to human Ionotropic glutamate receptor 2 | Homo sapiens | 1 | ALA1139549 | single protein format | Scientific Literature | |
9. | ALA829051 | B | Inhibition of [3H]-AMPA binding to human GluR2 receptors expressed in HEK 293 cells | Homo sapiens | 6 | ALA1139549 | cell-based format | Scientific Literature | |
10. | ALA863280 | F | Inhibitory effect on glutamate-induced calcium influx at homomeric human GLUA2 receptor expressed in HEK293 cells up to 300 uM | Homo sapiens | 1 | ALA1141230 | cell-based format | Scientific Literature | |
11. | ALA865009 | F | Inhibition of glutamate-induced calcium influx in HEK293 cells expressing human GLUA2 up to 100 uM | Homo sapiens | 1 | ALA1146072 | cell-based format | Scientific Literature | |
12. | ALA865015 | F | Inhibition of glutamate-induced calcium influx in HEK293 cells expressing human GLUA2 | Homo sapiens | 1 | ALA1146072 | cell-based format | Scientific Literature | |
13. | ALA871564 | F | Activity against human GLUR2 flip expressed in HEK293 cells assessed as glutamate-stimulated calcium influx by FLIPR assay | Homo sapiens | 20 | ALA1146878 | cell-based format | Scientific Literature | |
14. | ALA871565 | F | Activity against human GLUR2 flop expressed in HEK293 cells assessed as glutamate-stimulated calcium influx by FLIPR assay | Homo sapiens | 20 | ALA1146878 | cell-based format | Scientific Literature | |
15. | ALA856920 | F | Activity at human recombinant iGluR2 flip expressed in HEK293 cells measured as change in intracellular calcium ion concentration in presence of glutamate by FLIPR assay | Homo sapiens | 25 | ALA1146909 | cell-based format | Scientific Literature | |
16. | ALA856924 | F | Activity at human recombinant iGluR2 flop expressed in HEK293 cells measured as change in intracellular calcium ion concentration in presence of glutamate by FLIPR assay | Homo sapiens | 25 | ALA1146909 | cell-based format | Scientific Literature | |
17. | ALA914410 | F | Antagonist activity at human recombinant GLUA2-AMPA receptor expressed in HEK293 cells assessed as inhibition of glutamate-stimulated calcium influx by FLIPR assay | Homo sapiens | 5 | ALA1142988 | cell-based format | Scientific Literature | |
18. | ALA895664 | F | Agonist activity at GluR2Q expressed in HEK293 cells by Fluo-4/Ca2+ assay | 6 | ALA1148746 | cell-based format | Scientific Literature | ||
19. | ALA895665 | F | Agonist activity at GluR2Q expressed in HEK293 cells relative to S-Glutamate by Fluo-4/Ca2+ assay | 4 | ALA1148746 | cell-based format | Scientific Literature | ||
20. | ALA934441 | B | Binding affinity at iGluR2 receptor S1S2J domain expressed in sf9 cells by radioligand binding assay | 2 | ALA1143163 | cell-based format | Scientific Literature |