# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA837040 | F | Fold activation of estrogen-related receptor beta at 3 uM in cell-based reporter gene assay | 1 | ALA1141994 | cell-based format | Scientific Literature | ||
2. | ALA837153 | F | Fold activation of estrogen-related receptor beta at 10 uM in cell-based reporter gene assay | 1 | ALA1141994 | cell-based format | Scientific Literature | ||
3. | ALA837154 | F | Fold activation of estrogen-related receptor beta at 30 uM in cell-based reporter gene assay | 1 | ALA1141994 | cell-based format | Scientific Literature | ||
4. | ALA837727 | F | Fold activation of estrogen-related receptor beta at 100 nM in cell-based reporter gene assay | 1 | ALA1141994 | cell-based format | Scientific Literature | ||
5. | ALA860922 | B | Binding affinity to human ERbeta relative to estradiol by radiometric binding assay | Homo sapiens | 24 | ALA1146101 | single protein format | Scientific Literature | |
6. | ALA888442 | B | Binding affinity to ERbeta | Homo sapiens | 1 | ALA1145402 | single protein format | Scientific Literature | |
7. | ALA886439 | B | Inhibition of human ERbeta | Homo sapiens | 21 | ALA1139966 | single protein format | Scientific Literature | |
8. | ALA949846 | F | Antagonist activity at ERRbeta expressed in african green monkey CV1 cells by luciferase reporter gene assay | 1 | ALA1140941 | cell-based format | Scientific Literature | ||
9. | ALA972354 | B | Displacement of [3H]estradiol from human ERbeta receptor at 1 uM by radiometric binding assay | Homo sapiens | 1 | ALA1150267 | single protein format | Scientific Literature | |
10. | ALA1679772 | F | Agonist activity at ZFP-fused ERRbeta LBD expressed in HEK293 cells by TR-FRET assay | 2 | ALA1671812 | cell-based format | Scientific Literature | ||
11. | ALA1679773 | F | Agonist activity at ZFP-fused ERRbeta LBD expressed in HEK293 cells by TR-FRET assay relative to control | 1 | ALA1671812 | cell-based format | Scientific Literature | ||
12. | ALA1918212 | F | Agonist activity at ERRbeta expressed in human 293FT cells assessed as increase of transcriptional activity at 10 uM after 24 hrs by dual luciferase reporter gene assay | Homo sapiens | 1 | ALA1914388 | cell-based format | Scientific Literature | |
13. | ALA1961858 | B | Effect on ERR2(NR3B2) dependent reporter activity in HEK293 cells at 20 uM | 2 | ALA1961794 | cell-based format | Scientific Literature | ||
14. | ALA2330133 | B | Displacement of [3H]E2 from human recombinant ERbeta receptor after overnight incubation by liquid scintillation counting analysis relative to 17beta-estradiol | Homo sapiens | 9 | ALA2321717 | single protein format | Scientific Literature | |
15. | ALA2330135 | B | Displacement of [3H]E2 from human recombinant ERbeta receptor after overnight incubation by liquid scintillation counting analysis | Homo sapiens | 10 | ALA2321717 | single protein format | Scientific Literature | |
16. | ALA3635230 | B | Transactivation of ERRbeta (unknown origin) transfected in human HepG2 cells at 10 uM after 18 hrs by luciferase reporter assay relative to 17beta-estradiol | Homo sapiens | 3 | ALA3632562 | cell-based format | Scientific Literature | |
17. | ALA3635232 | B | Antagonist activity at ERRbeta (unknown origin) transfected in human HepG2 cells assessed as inhibition of genistein-induced effect at 50 uM after 18 hrs by luciferase reporter assay | Homo sapiens | 3 | ALA3632562 | cell-based format | Scientific Literature | |
18. | ALA3857090 | B | Inhibition of fluorescien-conjugated coactivator PGC1a binding to ERRbeta (unknown origin) after 1 hr by TR-FRET assay | Homo sapiens | 8 | ALA3856205 | single protein format | Scientific Literature | |
19. | ALA3999513 | B | Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as decrease in receptor transcriptional activity after 45 hrs by luciferase reporter gene assay | Homo sapiens | 13 | ALA3997814 | cell-based format | Scientific Literature | |
20. | ALA4131420 | B | Antagonist activity at recombinant GST-tagged human ERRbeta LBD assessed as inhibition of fluorescein-labeled coactivator peptide recruitment preincubated with enzyme followed by coactivator addition by LanthaScreen TR-FRET assay | Homo sapiens | 2 | ALA4130359 | single protein format | Scientific Literature |