# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA879065 | B | Inhibition of recombinant prenyl protein-specific protease Rce1 expressed in Sf9 cells at 10 uM | Homo sapiens | 2 | ALA1134177 | cell-based format | Scientific Literature | |
2. | ALA800857 | B | Inhibition of recombinant prenyl protein-specific protease Rcel expressed in Sf9 cells | Homo sapiens | 1 | ALA1134177 | cell-based format | Scientific Literature | |
3. | ALA800858 | B | Inhibition of recombinant prenyl protein-specific protease Rce1 in Sf9 cells at a concentration of 10 uM | Homo sapiens | 13 | ALA1134177 | cell-based format | Scientific Literature | |
4. | ALA1055573 | B | Inhibition of human RCE1 | Homo sapiens | 4 | ALA1152967 | single protein format | Scientific Literature | |
5. | ALA1794354 | B | PUBCHEM_BIOASSAY: Human Ras-Converting Enzyme Inhibition Assay Measured in Biochemical System Using Plate Reader - 2034-04_Inhibitor_Dose_DryPowder_Activity. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID2618] | 6 | ALA1201862 | biochemical format | PubChem BioAssays | ||
6. | ALA1794566 | B | PUBCHEM_BIOASSAY: Human Ras-Converting Enzyme Inhibition Assay Measured in Biochemical System Using Plate Reader - 2034-04_Inhibitor_Dose_CherryPick_Activity. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID2618] | 215 | ALA1201862 | biochemical format | PubChem BioAssays | ||
7. | ALA3742597 | B | Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residual activity at 10 uM measured every 30 to 60 seconds for 60 mins | Homo sapiens | 58 | ALA3739299 | single protein format | Scientific Literature | |
8. | ALA3742598 | B | Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residual activity measured every 30 to 60 seconds for 60 mins | Homo sapiens | 58 | ALA3739299 | single protein format | Scientific Literature | |
9. | ALA3742600 | B | Inhibition of Rce1 in human HCT116 cells assessed as mislocalization of EGFP-H-Ras in plasma membrane at 25 uM after 24 hrs by fluorescence assay | Homo sapiens | 1 | ALA3739299 | cell-based format | Scientific Literature | |
10. | ALA3742601 | B | Inhibition of Rce1 in human HCT116 cells assessed as mislocalization of EGFP-N-Ras in plasma membrane at 25 uM after 24 hrs by fluorescence assay | Homo sapiens | 1 | ALA3739299 | cell-based format | Scientific Literature | |
11. | ALA3742602 | B | Inhibition of Rce1 in human HCT116 cells assessed as mislocalization of EGFP-K-Ras in plasma membrane at 25 uM after 24 hrs by fluorescence assay | Homo sapiens | 5 | ALA3739299 | cell-based format | Scientific Literature | |
12. | ALA4360191 | A | Inhibition of Rce1 in human PC3 cells at 10 uM using KSKTKC(f)VI as substrate measured after 24 hrs by LC-MS/MS analysis | Homo sapiens | 1 | ALA4359814 | cell-based format | Scientific Literature |