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# Aladdin ID Assay Type Description Organism Compounds Reference BAO Format Source 1. ALA692999 B Maximum response (E max) against H1 receptor in rat aorta 1 tissue-based format Scientific Literature 2. ALA693000 B Relative potency against H1 receptor in rat aorta 1 tissue-based format Scientific Literature 3. ALA857125 F Compound was evaluated for mepyramine antagonism effects in rat aorta (relaxation) at a mepyramine concentration of 100 nM 1 tissue-based format Scientific Literature 4. ALA693636 B Effective concentration against histamine H1 receptor in rat aorta 1 tissue-based format Scientific Literature 5. ALA693637 B Compound was evaluated for binding activity against [3H]pyrilamine as radioligand for Histamine H1 receptor 1 single protein format Scientific Literature 6. ALA693638 F Effective concentration for agonism activity in relaxed rat aortic rings with intact endothelium, submaximally precontracted with 15.8 nM U-46,619; ND id no data 1 tissue-based format Scientific Literature 7. ALA693639 F Effective concentration for agonism activity in relaxed rat aortic rings with intact endothelium, submaximally precontracted with 15.8 nM U-46,619; ND is no data 1 tissue-based format Scientific Literature 8. ALA693640 F Intrinsic activity of the histamine as reported in relaxed rat aortic rings with intact endothelium, submaximally precontracted with 15.8 nM U-46,619 1 tissue-based format Scientific Literature 9. ALA693641 B Maximum response (E max) against H1 receptor in rat aorta 3 tissue-based format Scientific Literature 10. ALA693642 B Maximum response (E max) against Histamine H1 receptor endothelium-Denuded rings of guinea pig Aorta 1 single protein format Scientific Literature 11. ALA693643 B Relative potency against Histamine H1 receptor in endothelium-Denuded rings of guinea pig Aorta 1 tissue-based format Scientific Literature 12. ALA693644 F The compound was evaluated for intrinsic activity i.e. maximum histamine controls relative to contraction evoked by 10 uM PGF2-alpha in in relaxed rat aortic rings 1 tissue-based format Scientific Literature 13. ALA693645 F The compound was evaluated for intrinsic activity i.e. maximum histamine controls relative to contraction evoked by 10 uM PGF2-alpha in relaxed rat aortic rings 1 tissue-based format Scientific Literature 14. ALA693646 F The compound was evaluated for intrinsic activity in relaxed rat aortic rings with intact endothelium, submaximally precontracted with 15.8 nM U-46,619 5 tissue-based format Scientific Literature 15. ALA693647 F maximum relaxation evoked by carbachol in relaxed rat aortic rings with intact endothelium, submaximally precontracted with 15.8 nM U-46,619 1 tissue-based format Scientific Literature 16. ALA692701 B Binding affinity against Histamine H1 receptor was measured using radioligand ([3H]pyrilamine) binding assay 1 single protein format Scientific Literature 17. ALA692702 B Compound tested for its inhibitory activity against Histamine H1 receptor 7 single protein format Scientific Literature 18. ALA692703 B Binding affinity towards histamine H1 receptor from rat brain membranes using [3H]mepyramine as radioligand 6 assay format Scientific Literature 19. ALA692704 B Binding affinity towards histamine H1 receptor from rat brain membranes using [3H]mepyramine as radioligand; Not tested 10 assay format Scientific Literature 20. ALA692705 B Inhibitory binding of [3H]mepyramine to histamine H1 receptors in rat brain membranes 4 cell membrane format Scientific Literature