# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA698650 | F | In vivo agonist activity against histamine H2-receptor in lumen-perfused stomach of atropinized (1 mg/kg) anesthetized rat gastric secretion | 2 | organism-based format | Scientific Literature | |||
2. | ALA698651 | F | In vivo agonist activity against histamine H2-receptor in lumen-perfused stomach of atropinized (1 mg/kg) anesthetized rat gastric secretion at 128 ug/kg; -ve | 1 | organism-based format | Scientific Literature | |||
3. | ALA698652 | F | In vivo agonist activity against histamine H2-receptor in lumen-perfused stomach of atropinized (1 mg/kg) anesthetized rat gastric secretion at 187 ug/kg; -ve | 1 | organism-based format | Scientific Literature | |||
4. | ALA698653 | F | In vivo agonist activity against histamine H2-receptor in lumen-perfused stomach of atropinized (1 mg/kg) anesthetized rat gastric secretion at 256 ug/kg; -ve | 1 | organism-based format | Scientific Literature | |||
5. | ALA698654 | F | In vivo agonist activity against histamine H2-receptor in lumen-perfused stomach of atropinized (1 mg/kg) anesthetized rat gastric secretion at 512 ug/kg; -ve | 1 | organism-based format | Scientific Literature | |||
6. | ALA698655 | F | In vivo agonist activity against histamine H2-receptor in lumen-perfused stomach of atropinized (1 mg/kg) anesthetized rat gastric secretion at 64 ug/kg; -ve | 1 | organism-based format | Scientific Literature | |||
7. | ALA698656 | F | In vivo antagonist activity against histamine H2-receptor in lumen-perfused stomach of atropinized (1 mg/kg) anesthetized rat gastric secretion at 128 ug/kg; -ve | 4 | organism-based format | Scientific Literature | |||
8. | ALA698657 | F | In vivo antagonist activity against histamine H2-receptor in lumen-perfused stomach of atropinized (1 mg/kg) anesthetized rat gastric secretion at 187 ug/kg; weak inhibition | 1 | organism-based format | Scientific Literature | |||
9. | ALA698658 | F | In vivo antagonist activity against histamine H2-receptor in lumen-perfused stomach of atropinized (1 mg/kg) anesthetized rat gastric secretion at 256 ug/kg; -ve | 1 | organism-based format | Scientific Literature | |||
10. | ALA698812 | F | In vivo antagonist activity against histamine H2-receptor in lumen-perfused stomach of atropinized (1 mg/kg) anesthetized rat gastric secretion at 512 ug/kg; -ve | 1 | organism-based format | Scientific Literature | |||
11. | ALA857126 | F | Antagonistic activity for inhibition of histamine H2 receptor from anesthetized rats | 29 | assay format | Scientific Literature | |||
12. | ALA698813 | F | Antagonistic activity by inhibition histamine H2 receptor from rats. | 17 | assay format | Scientific Literature | |||
13. | ALA698814 | B | Affinity to the Histamine H2 receptor was determined expressed in CHO cell using [125I]iodoaminopotentidine as radioligand | 3 | cell-based format | Scientific Literature | |||
14. | ALA698815 | B | Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitro | 23 | single protein format | Scientific Literature | |||
15. | ALA698816 | B | Inhibitory activity against binding of [125I]-(Nle11)-HG-13 to Histamine H2 receptor in vitro; ND = Not determined | Rattus norvegicus | 2 | single protein format | Scientific Literature | ||
16. | ALA698818 | B | Competitive binding at Histamine H2 receptor at 10 uM; NA means compound failed to compete | Rattus norvegicus | 1 | single protein format | Scientific Literature | ||
17. | ALA698819 | B | Ability to displace [3H]tiotidine from histamine-H2 receptor at concentration of 10e-5 M | 1 | single protein format | Scientific Literature | |||
18. | ALA698992 | B | Ability to displace [3H]tiotidine from histamine-H2 receptor at concentration of 10e-7 M | 1 | single protein format | Scientific Literature | |||
19. | ALA697093 | B | Inhibition of H2 histamine receptor binding at a concentration of 10 uM; Showed negligible activities | 1 | single protein format | Scientific Literature | |||
20. | ALA868974 | B | Inhibition of rat histamine H2 receptor at 1 uM | Rattus norvegicus | 2 | single protein format | Scientific Literature |