| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA681450 | F | Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human GAT-1 transporter | 5 | assay format | Scientific Literature | |||
| 2. | ALA806333 | B | Inhibitory activity against human GABA transporter-1 (hGAT1) | 28 | single protein format | Scientific Literature | |||
| 3. | ALA881972 | B | Percent inhibition against GABA transporter at a compound concentration of 1 uM | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 4. | ALA862288 | B | Inhibition of GAT1 transport activity | Homo sapiens | 22 | single protein format | Scientific Literature | ||
| 5. | ALA1663477 | B | Inhibition of [3H]GABA uptake at GAT1 expressed in HEK cells | 18 | cell-based format | Scientific Literature | |||
| 6. | ALA1663478 | B | Inhibition of [3H]GABA uptake at GAT1 expressed in HEK cells at 100 uM | 1 | cell-based format | Scientific Literature | |||
| 7. | ALA1166723 | B | Binding affinity to GAT1 | 3 | single protein format | Scientific Literature | |||
| 8. | ALA1647445 | B | Displacement of [3H]Tiagabine from human recombinant GAT1 expressed in HEK293 cells by equilibrium binding assay | Homo sapiens | 52 | cell-based format | Scientific Literature | ||
| 9. | ALA1776005 | B | Inhibition of human GAT1-mediated GABA uptake | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 10. | ALA1918360 | B | Inhibition of human GAT1 assessed as [3H]GABA uptake | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 11. | ALA2208544 | B | Inhibition of human GAT1 expressed in tcA201 cells assessed as inhibition of [3H]GABA uptake at 1 mM after 3 mins by scintillation counting | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 12. | ALA2405421 | B | Inhibition of GABA uptake at GAT-1 (unknown origin) | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 13. | ALA2417030 | B | Inhibition of human GAT1 transfected in CHO cells assessed as [3H]GABA uptake after 20 mins by liquid scintillation counting analysis | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
| 14. | ALA2417034 | B | Inhibition of human GAT1 transfected in CHO cells assessed as [3H]GABA uptake at 100 uM after 20 mins by liquid scintillation counting analysis | Homo sapiens | 8 | cell-based format | Scientific Literature | ||
| 15. | ALA2432985 | B | Activity at GAT1 (unknown origin) expressed in african green monkey COS7 cells assessed as GABA release at 0.5 to 500 uM after 10 mins using [3H]-GABA pretreated for 1 hr before compound addition followed by wash out by reversed transport efflux assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 16. | ALA2432988 | B | Allosteric modulation of GAT-1 (unknown origin) expressed in african green monkey COS7 cells using [3H]-GABA as substrate at 20 uM | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 17. | ALA2432991 | B | Non-competitive inhibition of GAT-1 (unknown origin) expressed in african green monkey COS7 cells using [3H]-GABA as substrate | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 18. | ALA2433117 | B | Inhibition of GAT-1 (unknown origin) | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 19. | ALA2433118 | B | Inhibition of GAT-1 (unknown origin) expressed in african green monkey COS7 cells using [3H]-GABA as substrate after 10 mins by scintillation counting | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 20. | ALA3363226 | B | Inhibition of human GAT1 transfected in CHO cells assessed as [3H]GABA uptake after 20 mins by liquid scintillation counting analysis | Homo sapiens | 4 | cell-based format | Scientific Literature |
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