| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA696454 | B | Inhibition constant was evaluated against Histamine N-methyl-transferase | Cavia porcellus | 2 | ALA1122976 | single protein format | Scientific Literature | |
| 2. | ALA696455 | B | Inhibition constant was evaluated against Histamine N-methyl-transferase; ND is not determined | Cavia porcellus | 1 | ALA1122976 | single protein format | Scientific Literature | |
| 3. | ALA991565 | B | Inhibition of histamine N-methyl-transferase | 4 | ALA1144223 | single protein format | Scientific Literature | ||
| 4. | ALA2059994 | B | Inhibition of histamine N-methyltransferase by radiochemical assay | Homo sapiens | 1 | ALA2057181 | single protein format | Scientific Literature | |
| 5. | ALA2217166 | B | Binding affinity to HNMT in human HepG2 cell lysate after 1 hr by capture compound based LC/MS analysis | Homo sapiens | 1 | ALA2216748 | cell-based format | Scientific Literature | |
| 6. | ALA2217173 | B | Displacement of 3-(1-methyl-N-(pyridin-2-yl)-2-((4-(N-((S)-6,9,25-trioxo-29-((3aS,4S,6aR)-2-oxohexahydro-1H-thieno[3,4-d]imidazol-4-yl)-8-(4-(3-(trifluoromethyl)-3H-diazirin-3-yl)benzamido)-14,17,20-trioxa-5,10,24-triazanonacosyl)carbamimidoyl)phenylamino)methyl)-1H-benzo[d]imidazole-5-carboxamido)propanoic acid from HNMT in human HepG2 cell lysate after 1 hr by capture compound based LC/MS analysis | Homo sapiens | 1 | ALA2216748 | cell-based format | Scientific Literature | |
| 7. | ALA2217180 | B | Binding affinity to HNMT in human K562 cell lysate after 1 hr by capture compound based LC/MS analysis | Homo sapiens | 1 | ALA2216748 | cell-based format | Scientific Literature | |
| 8. | ALA4416340 | A | Inhibition of human HNMT expressed in Escherichia coli at 10 uM assessed as reduction in SAH level using histamine as substrate in presence of SAM incubated for 15 mins by LC-MS/MS analysis relative to control | Homo sapiens | 1 | ALA4414609 | assay format | Scientific Literature | |
| 9. | ALA4416347 | A | Inhibition of human HNMT expressed in Escherichia coli at 1 uM assessed as reduction in SAH level using histamine as substrate in presence of SAM incubated for 15 mins by LC-MS/MS analysis relative to control | Homo sapiens | 1 | ALA4414609 | assay format | Scientific Literature |
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