| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA771325 | B | Evaluated for the inhibition of Human leukocyte Proteinase 3 (PR-3) following a 10-min incubation with a 50-fold excess of inhibitor | 2 | ALA1125156 | single protein format | Scientific Literature | ||
| 2. | ALA771967 | B | Evaluated for the inhibition of Human leukocyte Proteinase 3 (PR-3) | 10 | ALA1125156 | single protein format | Scientific Literature | ||
| 3. | ALA771968 | B | Evaluated for the inhibition of Human leukocyte Proteinase 3 (PR-3); Inactivation was too fast to measure by sampling techniques | 2 | ALA1125156 | single protein format | Scientific Literature | ||
| 4. | ALA771969 | B | Evaluated for the inhibition of Human leukocyte Proteinase 3 (PR-3); Inactive | 2 | ALA1125156 | single protein format | Scientific Literature | ||
| 5. | ALA878681 | B | Compound was evaluated for inhibitory activity against Proteinase 3 | 1 | ALA1130769 | single protein format | Scientific Literature | ||
| 6. | ALA929935 | B | Ratio of Kinact to KI for human PR3 | Homo sapiens | 8 | ALA1143175 | single protein format | Scientific Literature | |
| 7. | ALA972416 | B | Inhibition of human PR3 at inhibitor to enzyme ratio of 500 after 30 mins | Homo sapiens | 9 | ALA1136882 | single protein format | Scientific Literature | |
| 8. | ALA1004879 | B | Inhibition of proteinase-3 in human U937 cells | Homo sapiens | 2 | ALA1156470 | cell-based format | Scientific Literature | |
| 9. | ALA1047944 | B | Inhibition of human proteinase 3 at 10 uM | Homo sapiens | 1 | ALA1156756 | single protein format | Scientific Literature | |
| 10. | ALA1047945 | B | Inhibition of human proteinase 3 at 60 uM | Homo sapiens | 1 | ALA1156756 | single protein format | Scientific Literature | |
| 11. | ALA1047946 | B | Inhibition of human proteinase 3 | Homo sapiens | 26 | ALA1156756 | single protein format | Scientific Literature | |
| 12. | ALA1065212 | B | Inhibition of human neutrophil proteinase 3 | Homo sapiens | 9 | ALA1156838 | single protein format | Scientific Literature | |
| 13. | ALA1113182 | B | Inhibition of human Proteinase-3 | Homo sapiens | 1 | ALA1154218 | single protein format | Scientific Literature | |
| 14. | ALA1228538 | B | Inhibition of human neutrophil proteinase 3 assessed as residual activity at 8.62 | Homo sapiens | 16 | ALA1221393 | single protein format | Scientific Literature | |
| 15. | ALA1771829 | B | Inhibition of proteinase 3 after 30 mins | 1 | ALA1770148 | single protein format | Scientific Literature | ||
| 16. | ALA2034576 | B | Inhibition of proteinase 3 using N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide as substrate after 60 mins | 10 | ALA2029305 | single protein format | Scientific Literature | ||
| 17. | ALA3095811 | B | Inhibition of human proteinase 3 using N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide as substrate measured for 30 mins by spectrophotometry | Homo sapiens | 4 | ALA3091365 | single protein format | Scientific Literature | |
| 18. | ALA3222424 | B | Inhibition of proteinase 3 in human neutrophil using N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide as chromogenic substrate measured for 60 mins by chromogenic assay | Homo sapiens | 2 | ALA3217450 | single protein format | Scientific Literature | |
| 19. | ALA3371653 | B | Inhibition of human PR3 using N-EY-FRET as substrate after 20 mins by fluorescence assay | Homo sapiens | 4 | ALA3351424 | single protein format | Scientific Literature | |
| 20. | ALA3371655 | B | Inhibition of human PR3 using N-EY-FRET as substrate at 6 uM after 20 mins by fluorescence assay | Homo sapiens | 1 | ALA3351424 | single protein format | Scientific Literature |
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