| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA979922 | F | Agonist activity at rat recombinant GABAA alpha-4-beta-3-gamma-2 receptor expressed in HEK293 cells assessed as induction of current by whole cell patch-clamp technique | Rattus norvegicus | 1 | cell-based format | Scientific Literature | ||
| 2. | ALA979927 | F | Antagonist activity at recombinant rat GABAA alpha-4-beta-3-gamma-2 receptor expressed in HEK293 cells assessed as inhibition of GABA-induced current at 1 mM by whole-cell patch-clamp technique | Rattus norvegicus | 1 | cell-based format | Scientific Literature | ||
| 3. | ALA979931 | B | Intrinsic activity at recombinant rat GABAA alpha-4-beta-3-gamma-2 receptor expressed in HEK293 cells assessed as induction of current at 1 mM by whole-cell patch-clamp technique relative to GABA | Rattus norvegicus | 2 | cell-based format | Scientific Literature | ||
| 4. | ALA971711 | F | Agonist activity at recombinant rat GABAA alpha-4-beta-3-gamma-2 receptor expressed in HEK293 cells assessed as potentiation of GABA-induced current at 1 mM by whole-cell patch-clamp technique | Rattus norvegicus | 1 | cell-based format | Scientific Literature | ||
| 5. | ALA971726 | F | Agonist activity at rat recombinant GABAA alpha-4-beta-3-gamma-2 receptor expressed in HEK293 cells assessed as normalization of GABA-induced current by whole cell patch-clamp technique | Rattus norvegicus | 1 | cell-based format | Scientific Literature | ||
| 6. | ALA3888612 | B | [35S]-TBPS Displacement Assay: The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors. | 18 | single protein format | BindingDB Database |
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