| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA652602 | F | Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human BGT-1 transporter | 5 | assay format | Scientific Literature | |||
| 2. | ALA806334 | B | Inhibition of human GABA transporter (hBGT-1) activity. | 22 | single protein format | Scientific Literature | |||
| 3. | ALA806335 | B | Compound was evaluated for inhibitory activity against human GABA transporter (hBGT-1) at 100 uM concentration | 1 | single protein format | Scientific Literature | |||
| 4. | ALA806336 | B | Compound was evaluated for inhibitory activity against human GABA transporter (hBGT-1)at 100 uM concentration | 5 | single protein format | Scientific Literature | |||
| 5. | ALA1809624 | B | Inhibition of GABA transporter at 4 uM | 1 | single protein format | Scientific Literature | |||
| 6. | ALA1918362 | B | Inhibition of human BGT1 assessed as [3H]GABA uptake | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 7. | ALA1166725 | B | Binding affinity to BGT-1 | 1 | single protein format | Scientific Literature | |||
| 8. | ALA1647450 | B | Inhibition of BGT1 | 1 | single protein format | Scientific Literature | |||
| 9. | ALA1776006 | B | Inhibition of human BGT1-mediated GABA uptake at 100 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 10. | ALA2208545 | B | Inhibition of human BGT1 expressed in tcA201 cells assessed as inhibition of [3H]GABA uptake at 1 mM after 3 mins by scintillation counting | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 11. | ALA2213048 | B | Inhibition of GABA transporter at 10 uM by CEREP assay | 1 | single protein format | Scientific Literature | |||
| 12. | ALA2417027 | B | Inhibition of human BGT1 transfected in CHO cells assessed as [3H]GABA uptake after 20 mins by liquid scintillation counting analysis | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 13. | ALA2417031 | B | Inhibition of human BGT1 transfected in CHO cells assessed as [3H]GABA uptake at 100 uM after 20 mins by liquid scintillation counting analysis | Homo sapiens | 8 | cell-based format | Scientific Literature | ||
| 14. | ALA3363499 | B | Inhibition of human BGT1 transfected in CHO cells assessed as [3H]GABA uptake after 20 mins by liquid scintillation counting analysis | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 15. | ALA3363501 | B | Inhibition of human BGT1 transfected in CHO cells assessed as [3H]GABA uptake at 100 uM after 20 mins by liquid scintillation counting analysis | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 16. | ALA3877714 | B | Inhibition of human BGT-1 expressed in thymidine kinase deficient mouse LM cells assessed as decrease in [3H]GABA uptake after 10 mins by scintillation counter method | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 17. | ALA4031697 | B | Inhibition of human BGT1 expresses in tsA201 cells assessed as reduction in [3H]GABA uptake after 3 mins by scintillation counting method | Homo sapiens | 33 | cell-based format | Scientific Literature | ||
| 18. | ALA4031712 | B | Inhibition of human BGT1 F295Y mutant expressed in tsA201 cells assessed as reduction in [3H]GABA uptake after 3 mins by scintillation counting method | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 19. | ALA4031713 | B | Inhibition of human BGT1 Q299L mutant expressed in tsA201 cells assessed as reduction in [3H]GABA uptake after 3 mins by scintillation counting method | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 20. | ALA4031714 | B | Inhibition of human BGT1 K310N mutant expressed in tsA201 cells assessed as reduction in [3H]GABA uptake after 3 mins by scintillation counting method | Homo sapiens | 3 | cell-based format | Scientific Literature |
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