# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA2091159 | B | Inhibition of thrombin activated human TG3 by fluorescent transamidation assay | Homo sapiens | 69 | ALA2086255 | single protein format | Scientific Literature | |
2. | ALA2155211 | B | Inhibition of human TGM3 | Homo sapiens | 1 | ALA2150866 | single protein format | Scientific Literature | |
3. | ALA2214884 | B | Inhibition of transglutaminase 3 | 4 | ALA2203174 | single protein format | Scientific Literature | ||
4. | ALA3388937 | B | Inhibition of human transglutaminase 3 using ((benzyloxy)carbonyl)-L-glutaminyl-L-serine peptide substrate assessed as Kinh/Ki ratio by GDH coupled assay | Homo sapiens | 8 | ALA3351998 | single protein format | Scientific Literature | |
5. | ALA4019587 | B | Inactivation of activated human TG3 assessed as rate constant of enzyme inactivation using FRET- quenched A101 as substrate by fluorescence assay | Homo sapiens | 2 | ALA4017513 | single protein format | Scientific Literature | |
6. | ALA4223777 | B | Irreversible inhibition of human TGase 3 assessed as ratio of Kinact/Ki using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assay | Homo sapiens | 3 | ALA4219231 | single protein format | Scientific Literature | |
7. | ALA5158934 | B | Inhibition of TG3 (unknown origin) using peptidic FRET quenched probe A101 as substrate and measured by fluorescence-based assay | Homo sapiens | 3 | ALA5154739 | single protein format | Scientific Literature | |
8. | ALA5233096 | B | Reversible inhibition of activated human TG3 using peptidic FRET-quenched probe A101 as substrate by fluorescence based assay relative to control | Homo sapiens | 4 | ALA5230175 | single protein format | Scientific Literature |