| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA615223 | B | In vitro inhibitory activity against human 11 beta hydroxysteroid dehydrogenase type 1 using scintillation proximity assay (SPA) | 3 | ALA1135754 | single protein format | Scientific Literature | ||
| 2. | ALA615226 | B | Ability to convert [3H]cortisol to the tritium labeled cortisone in the presence of human 11 beta hydroxysteroid dehydrogenase type 2 | 3 | ALA1135754 | single protein format | Scientific Literature | ||
| 3. | ALA832598 | B | Inhibitory concentration against human 11-beta-hydroxysteroid dehydrogenase 1 | Homo sapiens | 11 | ALA1139567 | single protein format | Scientific Literature | |
| 4. | ALA868712 | B | Inhibitory activity against human 11beta-HSD1 | Homo sapiens | 24 | ALA1141865 | single protein format | Scientific Literature | |
| 5. | ALA869368 | F | In vivo inhibition of 11beta-HSD1 at 4 hr (10 mg/kg, po) assessed by extent of cortisone to cortisol conversion | 13 | ALA1141865 | organism-based format | Scientific Literature | ||
| 6. | ALA869369 | F | In vivo inhibition of 11beta-HSD1 at 16 hr (10 mg/kg, po) assessed by extent of cortisone to cortisol conversion | 11 | ALA1141865 | organism-based format | Scientific Literature | ||
| 7. | ALA859753 | F | In vivo inhibition of 11beta-HSD1 at 1 h (10 mg/kg, po) assessed by extent of cortisone to cortisol conversion | 2 | ALA1141865 | organism-based format | Scientific Literature | ||
| 8. | ALA863120 | B | Inhibition of human recombinant 11-beta-HSD1 expressed in HEK293 cells | Homo sapiens | 7 | ALA1148531 | cell-based format | Scientific Literature | |
| 9. | ALA853210 | B | Inhibition of human recombinant 11-beta-HSD1 expressed in HEK293 cells at 10 uM | Homo sapiens | 7 | ALA1148531 | cell-based format | Scientific Literature | |
| 10. | ALA853223 | B | Inhibition of human recombinant 11-beta-HSD1 transfected in intact HEK293 cells | Homo sapiens | 7 | ALA1148531 | cell-based format | Scientific Literature | |
| 11. | ALA855991 | B | Inhibition of human 11beta-HSD1 | Homo sapiens | 17 | ALA1137282 | single protein format | Scientific Literature | |
| 12. | ALA855996 | B | Inhibition of human 11beta-HSD1 expressed in HEK cells | Homo sapiens | 17 | ALA1137282 | cell-based format | Scientific Literature | |
| 13. | ALA856010 | B | Inhibition of human 11beta-HSD1 expressed in Escherichia coli | Homo sapiens | 17 | ALA1137283 | assay format | Scientific Literature | |
| 14. | ALA906988 | B | Inhibition of human 11beta-HSD1 expressed in HEK293 cells | Homo sapiens | 17 | ALA1137283 | cell-based format | Scientific Literature | |
| 15. | ALA909895 | B | Inhibition of human 11beta-HSD1 expressed in Escherichia coli by SPA | Homo sapiens | 22 | ALA1139224 | assay format | Scientific Literature | |
| 16. | ALA909897 | B | Inhibition of human 11beta-HSD1 expressed in HEK293 cells by FPIA | Homo sapiens | 22 | ALA1139224 | cell-based format | Scientific Literature | |
| 17. | ALA856747 | B | Inhibition of human 11beta-HSD1 | Homo sapiens | 18 | ALA1139681 | single protein format | Scientific Literature | |
| 18. | ALA856751 | B | Inhibition of human 11beta-HSD1 expressed in HEK293 cells | Homo sapiens | 11 | ALA1139681 | cell-based format | Scientific Literature | |
| 19. | ALA907396 | B | Inhibition of human truncated 11beta-HSD1 assessed as inhibition of radiolabeled cortisone to cortisol conversion by SPA | Homo sapiens | 19 | ALA1145299 | single protein format | Scientific Literature | |
| 20. | ALA907400 | B | Inhibition of human 11beta-HSD1 expressed in HEK293 cells assessed as inhibition of cortisol formation by fluorescent polarization immunoassay | Homo sapiens | 19 | ALA1145299 | cell-based format | Scientific Literature |
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