| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3864103 | B | Inhibition of ppGalNAcT2 (unknown origin) in presence of OGT, EA2 and UDP-GlcNAc incubated for 25 mins at 37 degC | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 2. | ALA4386611 | B | Inhibition of catalytic activity of human recombinant FLAG-tagged ppGalNAcT2 expressed in HEK293T cells and using 5-FAM labelled-EA2 peptide as substrate incubated for 30 mins by HPLC-based enzyme assay | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
| 3. | ALA4386612 | B | Binding affinity of human recombinant FLAG-tagged ppGalNAcT2 expressed in HEK293 cells assessed as dissociation constant by SPR analysis | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 4. | ALA4386613 | B | Binding affinity of human recombinant FLAG-tagged ppGalNAcT2 expressed in HEK293 cells assessed as association rate by SPR analysis | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 5. | ALA4386614 | B | Binding affinity of human recombinant FLAG-tagged ppGalNAcT2 expressed in HEK293 cells assessed as dissociation rate by SPR analysis | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 6. | ALA4386615 | B | Competitive inhibition of human recombinant FLAG-tagged ppGalNAcT2 expressed in HEK293 cells using EA2 peptide as substrate by HPLC-based enzyme assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 7. | ALA4386616 | B | Non-competitive inhibition of human recombinant FLAG-tagged ppGalNAcT2 expressed in HEK293 cells using UDP-GalNAc as substrate by HPLC-based enzyme assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 8. | ALA4386624 | B | Inhibition of catalytic activity of human recombinant FLAG-tagged ppGalNAcT2 using Muc2 peptide as substrate incubated for 30 mins by HPLC-based enzyme assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 9. | ALA4386625 | B | Inhibition of catalytic activity of human recombinant FLAG-tagged ppGalNAcT2 using Muc5AC peptide as substrate incubated for 30 mins by HPLC-based enzyme assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 10. | ALA4386626 | B | Inhibition of catalytic activity of human recombinant FLAG-tagged ppGalNAcT2 using Muc7 peptide as substrate incubated for 30 mins by HPLC-based enzyme assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 11. | ALA4386627 | B | Inhibition of catalytic activity of human recombinant FLAG-tagged ppGalNAcT2 W282A mutant expressed in HEK293 cells using EA2 peptide as substrate by HPLC-based enzyme assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 12. | ALA4386629 | B | Inhibition of ppGalNAcT2 in human HT-29 cells assessed as reduction in O-GalNAc glycans by measuring PNA lectin signal on cell surface at 40 uM incubated for 48 hrs by DAPI staining based immunofluorescence method | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 13. | ALA4386630 | B | Inhibition of ppGalNAcT2 in human HT-29 cells assessed as reduction in O-GalNAc glycans by measuring VVA lectin expression at 20 to 60 uM incubated for 48 hrs by Western blot analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 14. | ALA4386631 | B | Inhibition of ppGalNAcT2 in human HT-29 cells assessed as reduction in O-GalNAc glycans by measuring PNA lectin expression at 20 to 60 uM incubated for 48 hrs by Western blot analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 15. | ALA4386649 | B | Inhibition of ppGalNAcT2 in human Jurkat cells assessed as reduction in O-GalNAc glycosylation by measuring VVA lectin expression at 40 uM incubated for 48 hrs by Western blot analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 16. | ALA4386650 | B | Inhibition of ppGalNAcT2 in human HCT116 cells assessed as reduction in O-GalNAc glycosylation by measuring VVA lectin expression at 40 uM incubated for 48 hrs by Western blot analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 17. | ALA4386651 | B | Inhibition of ppGalNAcT2 in human SW480 cells assessed as reduction in O-GalNAc glycosylation by measuring VVA lectin expression at 40 uM incubated for 48 hrs by Western blot analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 18. | ALA4386652 | B | Inhibition of ppGalNAcT2 in human RKO cells assessed as reduction in O-GalNAc glycosylation by measuring VVA lectin expression at 40 uM incubated for 48 hrs by Western blot analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 19. | ALA4386663 | B | Inhibition of ppGalNAcT2 in human HT-29 cells assessed as reduction in PDPN O-GalNAc glycosylation by at 40 uM incubated for 48 hrs by jacalin lectin based immunoprecipitation analysis | Homo sapiens | 1 | cell-based format | Scientific Literature |
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