| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA680696 | B | Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 1 | 5 | cell-based format | Scientific Literature | |||
| 2. | ALA680697 | B | Binding affinity for Excitatory amino acid transporter 1 (EAAT-1) in Glu uptake system | 11 | single protein format | Scientific Literature | |||
| 3. | ALA680702 | F | Potency (100 uM) to induce a transport current in the presence of glutamate in oocytes expressing human excitatory amino acid transporter 1 (EAAT1) | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
| 4. | ALA680703 | F | Potency (100 uM) to induce a transport current in the absence of glutamate in oocytes expressing human excitatory amino acid transporter 1 (EAAT1) | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
| 5. | ALA881962 | B | Inhibitory concentration against glutamate uptake in HEK cells expressing human Excitatory amino acid transporter 1 | Homo sapiens | 27 | cell-based format | Scientific Literature | ||
| 6. | ALA859747 | F | Binding affinity to human EAAT1 expressed in HEK293 cells in FMP (FLPR) assay | Homo sapiens | 12 | cell-based format | Scientific Literature | ||
| 7. | ALA870600 | B | Activity against human EAAT1 transfected in HEK293 cells | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 8. | ALA907700 | F | Inhibition of human EAAT1 expressed in HEK293 cells by FLIPR membrane potential assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 9. | ALA907705 | F | Substrate activity at human EAAT1 expressed in HEK293 cells by FLIPR membrane potential assay | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 10. | ALA907708 | F | Substrate activity at human EAAT1 expressed in HEK293 cells at 1000 uM relative to glutamate by FLIPR membrane potential assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 11. | ALA907711 | F | Substrate activity at human EAAT1 expressed in HEK293 cells relative to glutamate by FLIPR membrane potential assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 12. | ALA2067159 | B | Inhibition of human EAAT1 expressed in HEK293 cells assessed as inhibition of 3[H]-D-Aspartate uptake after 6 mins by scintillation counting method | Homo sapiens | 16 | cell-based format | Scientific Literature | ||
| 13. | ALA1016585 | B | Inhibition of glutamate-induced depolarization in human EAAT1 expressed in HEK293 cells by FMP assay | Homo sapiens | 12 | cell-based format | Scientific Literature | ||
| 14. | ALA1016590 | B | Inhibition of [3H]D-Asp uptake at EAAT1 in HEK293 cells | Homo sapiens | 11 | cell-based format | Scientific Literature | ||
| 15. | ALA998472 | B | Displacement of [3H]D-Asp from human EAAT1 receptor expressed in HEK293 cells | Homo sapiens | 28 | cell-based format | Scientific Literature | ||
| 16. | ALA998475 | B | Activity of human EAAT1 expressed in HEK293 cells up to 100 uM | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 17. | ALA998478 | B | Activity at human EAAT1 expressed in HEK293 cells assessed as inhibition of Glu-induced fluorescent response by FLIPR membrane potential blue assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 18. | ALA1261598 | B | Inhibition of human EAAT1 expressed in HEK293 cells by [3H]D-Asp uptake assay | Homo sapiens | 21 | cell-based format | Scientific Literature | ||
| 19. | ALA1919953 | B | Inhibition of EAAT1-mediated D-aspartate transport at 100 uM | 2 | single protein format | Scientific Literature | |||
| 20. | ALA2214981 | B | Inhibition of [3H]-D-aspartate uptake at human EAAT1 expressed in HEK293 cells after 6 mins by scintillation counting | Homo sapiens | 6 | cell-based format | Scientific Literature |
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