| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA656546 | B | Inhibition of binding of IL-8 to membranes of cloned CXC chemokine receptor 1 expressed in CHO Cells using [125I]IL-8 radioligand | Homo sapiens | 8 | assay format | Scientific Literature | ||
| 2. | ALA662152 | B | Displacement of [125I]IL-8 from CHO cell membrane expressing human CXCR1 receptor at a concentration of 20 uM | 5 | cell-based format | Scientific Literature | |||
| 3. | ALA828738 | B | Inhibitory concentration against interleukin-8 receptor of human neutrophils by using [125I]IL-8 (0.125 nM) as radioligand | Homo sapiens | 24 | single protein format | Scientific Literature | ||
| 4. | ALA828743 | B | Concentration required to inhibit [125I]-IL-8 binding towards C-X-C chemokine receptor type 1 of human expressed in CHO cells | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
| 5. | ALA828097 | B | Inhibition of C-X-C chemokine receptor type 1 | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 6. | ALA833463 | F | Inhibition of interleukin-8 induced elastase release from human neutrophils | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 7. | ALA863291 | B | Inhibitory activity against CXCR1(IL-8A) receptor by radioligand binding assay at 10 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 8. | ALA870520 | B | Inhibition of human CXCR1 at 10 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 9. | ALA912816 | B | Displacement of [125I]hCXCL8 from human CXCR1 receptor expressed in BaF3 cells | Homo sapiens | 13 | cell-based format | Scientific Literature | ||
| 10. | ALA853688 | B | Displacement of [125I]hCXCL8 from human CXCR1 receptor expressed in BaF3 cells at >10000 nM | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 11. | ALA908414 | B | Displacement of [125I]IL8 from CXCR1 expressed in CHO cells | Homo sapiens | 18 | cell-based format | Scientific Literature | ||
| 12. | ALA1805403 | B | Noncompetitive inhibition of human CXCR1 assessed as inhibition of CXCL8-induced neutrophile chemotaxis at 10 nM | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 13. | ALA927477 | B | Binding affinity to CXCR1 | 21 | single protein format | Scientific Literature | |||
| 14. | ALA927215 | B | Inhibition of CXCR1 | 37 | single protein format | Scientific Literature | |||
| 15. | ALA927218 | B | Inhibition of CXCR1-mediated chemotaxis in Ba/F3 cells expressing human CXCR1 | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 16. | ALA927220 | B | Inhibition of CXCR1 at >10000 nM | 4 | single protein format | Scientific Literature | |||
| 17. | ALA927219 | B | Inhibition of CXCR1-mediated chemotaxis in Ba/F3 cells expressing human CXCR1 at >10000 nM | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 18. | ALA928588 | B | Inhibition of CXCR1 upto 1 uM | 1 | single protein format | Scientific Literature | |||
| 19. | ALA1909127 | B | DRUGMATRIX: Chemokine CXCR1 (IL-8A) | 871 | single protein format | DrugMatrix | |||
| 20. | ALA1930406 | B | Inhibition of CXCR1 by Ca(2+) flux assay | 1 | single protein format | Scientific Literature |
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