# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1050833 | Binding | Selectivity for PRKCH as proportion of 290 kinases in screen with similar potency; non-selective = 1 highly selective = 0 | Homo sapiens | 1 | ALA1150977 | single protein format | Scientific Literature | |
2. | ALA1060261 | Binding | Binding constant for PRKCH kinase domain | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
3. | ALA1049983 | Binding | Inhibition of PRKCN at 2 uM | 1 | ALA1154644 | single protein format | Scientific Literature | ||
4. | ALA1056860 | Binding | Inhibition of PKCeta assessed as residual enzyme activity at 10 uM relative to untreated control | 4 | ALA1154186 | single protein format | Scientific Literature | ||
5. | ALA1057606 | Binding | Inhibition of PRKCH assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
6. | ALA1041406 | Binding | Inhibition of PKCeta at 1 uM | 1 | ALA1154622 | single protein format | Scientific Literature | ||
7. | ALA1037488 | Binding | Inhibition of PKCeta by IMAP kinase assay | 1 | ALA1155984 | single protein format | Scientific Literature | ||
8. | ALA1040277 | Binding | Residual activity of PKCeta at 1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
9. | ALA1070483 | Binding | Residual activity of PKCeta at 0.1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
10. | ALA1050340 | Binding | Residual activity of PKCeta at 10 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
11. | ALA1040090 | Binding | Inhibition of PKCeta by SPA | 10 | ALA1156112 | single protein format | Scientific Literature | ||
12. | ALA1039090 | Binding | Inhibition of PKCeta by IMAP kinase assay | 1 | ALA1156064 | single protein format | Scientific Literature | ||
13. | ALA1047195 | Binding | Inhibition of PKCeta by IMAP fluorescence polarization technology | 1 | ALA1156015 | single protein format | Scientific Literature | ||
14. | ALA1053590 | Binding | Inhibition of PKCeta at 1 uM | 1 | ALA1154027 | single protein format | Scientific Literature | ||
15. | ALA758469 | Binding | Inhibition of protein kinase C eta | Homo sapiens | 6 | ALA1129020 | single protein format | Scientific Literature | |
16. | ALA761875 | Binding | Inhibition of protein kinase C eta | 8 | ALA1129127 | single protein format | Scientific Literature | ||
17. | ALA772751 | Binding | Inhibition of Protein kinase C eta | 1 | ALA1148433 | single protein format | Scientific Literature | ||
18. | ALA770091 | Binding | Inhibition of Protein kinase C eta | Homo sapiens | 10 | ALA1129363 | single protein format | Scientific Literature | |
19. | ALA770092 | Binding | Inhibition of Protein kinase C eta expressed in Sf-9 cells | Homo sapiens | 13 | ALA1128824 | cell-based format | Scientific Literature | |
20. | ALA770093 | Binding | Inhibition of Protein kinase C eta expressed in Sf-9 cells (inactive) | Homo sapiens | 1 | ALA1128824 | cell-based format | Scientific Literature |