# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3427912 | Binding | Inhibition of human full length N-terminal GST-tagged PRK1 expressed in insect cells using glycogen synthase derived peptide as substrate at 100 nM by radiometric assay in presence of [32P]ATP | Homo sapiens | 1 | ALA3425434 | cell-based format | Scientific Literature | |
2. | ALA3630942 | Binding | Inhibition of PKN1 (unknown origin) at 10 uM after 120 mins P33 radiolabeled kinase activity assay | Homo sapiens | 3 | ALA3627608 | single protein format | Scientific Literature | |
3. | ALA3750016 | Binding | Inhibition of human PKN1 using [KKLNRTLSVA] as substrate | Homo sapiens | 1 | ALA3745707 | single protein format | Scientific Literature | |
4. | ALA3751062 | Binding | Inhibition of PRK1 (unknown origin) at 1 uM | Homo sapiens | 1 | ALA3745631 | single protein format | Scientific Literature | |
5. | ALA3749781 | Binding | Inhibition of PKN1 (unknown origin) | Homo sapiens | 1 | ALA3745712 | single protein format | Scientific Literature | |
6. | ALA3761170 | Binding | Inhibition of PRK1 (unknown origin) at 100 nM | Homo sapiens | 1 | ALA3758169 | single protein format | Scientific Literature | |
7. | ALA3790302 | Binding | Inhibition of PKN1 (unknown origin) in presence of [gamma33P]ATP | Homo sapiens | 4 | ALA3785066 | single protein format | Scientific Literature | |
8. | ALA3815963 | Binding | Inhibition of human PKN1 at 1 uM using [KKLNRTLSVA] as substrate | Homo sapiens | 1 | ALA3813650 | single protein format | Scientific Literature | |
9. | ALA3816512 | Binding | Inhibition of full length recombinant human GST-tagged PRK1 expressed in baculovirus expression system at 1 uM relative to control | Homo sapiens | 1 | ALA3813614 | assay format | Scientific Literature | |
10. | ALA3820668 | Binding | Inhibition of PKN1 (unknown origin) incubated for 1 hr by spectrophotometric analysis | Homo sapiens | 2 | ALA3817824 | single protein format | Scientific Literature | |
11. | ALA1071348 | Binding | Residual activity of PRK1 at 10 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
12. | ALA1100999 | Binding | Inhibition of PRK1 at 10 uM | 2 | ALA1154277 | single protein format | Scientific Literature | ||
13. | ALA1103221 | Binding | Inhibition of PKN1 at 5 uM | 1 | ALA1154316 | single protein format | Scientific Literature | ||
14. | ALA1108243 | Binding | Inhibition of PRK1 at 10 uM | 16 | ALA1157789 | single protein format | Scientific Literature | ||
15. | ALA1117734 | Binding | Inhibition of PKN1 at 10 uM | 1 | ALA1155477 | single protein format | Scientific Literature | ||
16. | ALA1166815 | Binding | Inhibition of PKN1 at 1 uM | 6 | ALA1165965 | single protein format | Scientific Literature | ||
17. | ALA1175223 | Binding | Inhibition of PKN1 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
18. | ALA1244251 | Binding | Inhibition of PRK1 at 1 uM after 60 mins by FRET assay in presence of 10 uM ATP | 7 | ALA1240340 | single protein format | Scientific Literature | ||
19. | ALA1244930 | Binding | Binding affinity to PKN1 | 7 | ALA1240346 | single protein format | Scientific Literature | ||
20. | ALA1252620 | Binding | Inhibition of PKN1 at 1 uM in presence of 10 uM ATP by Select Screen kinase assay relative to untreated control | 3 | ALA1250448 | single protein format | Scientific Literature |