| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA680875 | F | The potency at recombinant rat AMPA-R was measured on GluR4 receptor expressed in Xenopus Laevis oocytes | 1 | cell-based format | Scientific Literature | |||
| 2. | ALA680876 | B | Binding affinity towards GluR4 receptor from rat brain | 1 | assay format | Scientific Literature | |||
| 3. | ALA696663 | F | Effective concentration of compound was determined for electrophysiological properties on Ionotropic glutamate receptor AMPA 4 (GluR4) using rat cortical slice model in Xenopus laevis oocytes | 2 | cell-based format | Scientific Literature | |||
| 4. | ALA919619 | F | Antagonist activity at rat homomeric recombinant GluR4 expressed in HEK293 cells assessed as inhibition of intracellular calcium concentration by FLIPR assay | Rattus norvegicus | 6 | cell-based format | Scientific Literature | ||
| 5. | ALA919629 | F | Antagonist activity at rat homomeric recombinant GluR4 expressed in HEK293 cells assessed as inhibition of intracellular calcium concentration at 30 uM by FLIPR assay | Rattus norvegicus | 5 | cell-based format | Scientific Literature | ||
| 6. | ALA920256 | B | Displacement of [3H]AMPA from rat recombinant GluR4 expressed in Sf9 cells | Rattus norvegicus | 6 | cell-based format | Scientific Literature | ||
| 7. | ALA928078 | B | Activity at rat cloned iGluR4 expressed in human HEK293 cells by calcium imaging assay | Rattus norvegicus | 6 | cell-based format | Scientific Literature | ||
| 8. | ALA928079 | B | Activity at rat cloned iGluR4 expressed in human HEK293 cells by calcium imaging assay relative to L-glutamate | Rattus norvegicus | 5 | cell-based format | Scientific Literature | ||
| 9. | ALA1036611 | B | Inhibition of rat recombinant GluR4 expressed in Xenopus oocytes assessed as inhibition of kainate-induced evoked current at 3 uM by two electrode voltage clamp method | Rattus norvegicus | 1 | cell-based format | Scientific Literature | ||
| 10. | ALA1028970 | B | Displacement of (R,S)-[5-methyl-3H]AMPA from rat recombinant flop iGluR4 expressed in Sf9 cells | Rattus norvegicus | 17 | cell-based format | Scientific Literature | ||
| 11. | ALA1029769 | F | Agonist activity at cyclothiazide-desensitized rat recombinant flip iGluR4 expressed in Xenopus laevis oocytes by two electrode voltage-clamp electrophysiology method | Rattus norvegicus | 4 | cell-based format | Scientific Literature | ||
| 12. | ALA1029770 | F | Agonist activity at cyclothiazide-desensitized rat recombinant flop iGluR4c expressed in Xenopus laevis oocytes by two electrode voltage-clamp electrophysiology method | Rattus norvegicus | 1 | cell-based format | Scientific Literature | ||
| 13. | ALA1059438 | B | Displacement of [3H]AMPA from rat recombinant GluR4 flop isoform expressed in baculovirus infected Sf9 cells | Rattus norvegicus | 3 | cell-based format | Scientific Literature | ||
| 14. | ALA1059448 | F | Agonist activity at rat recombinant GluR4 flip isomer expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4/AM assay | Rattus norvegicus | 5 | cell-based format | Scientific Literature | ||
| 15. | ALA1059449 | F | Agonist activity at rat recombinant GluR4 flip isomer expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4/AM assay relative to glutamic acid | Rattus norvegicus | 4 | cell-based format | Scientific Literature | ||
| 16. | ALA1105525 | F | Agonist activity at rat recombinant GluA4 receptor flip isoform expressed in HEK293 cells assessed as effect on cyclothiazide-induced calcium flux by Fluo-4/AM staining-based fluorescence assay | Rattus norvegicus | 3 | cell-based format | Scientific Literature | ||
| 17. | ALA1106357 | F | Antagonist activity at rat recombinant GluA4 receptor flip isoform expressed in HEK293 cells assessed as effect on cyclothiazide-induced calcium flux by Fluo-4/AM staining-based fluorescence assay | Rattus norvegicus | 1 | cell-based format | Scientific Literature | ||
| 18. | ALA1108134 | B | Activity at rat recombinant GluA4 receptor flip isoform expressed in HEK293 cells assessed as potentiation of 3000 uM glutamate-induced current at 100 uM relative to control | Rattus norvegicus | 1 | cell-based format | Scientific Literature | ||
| 19. | ALA1108135 | B | Activity at rat recombinant GluA4 receptor flop isoform expressed in HEK293 cells assessed as potentiation of 3000 uM glutamate-induced current at 100 uM relative to control | Rattus norvegicus | 1 | cell-based format | Scientific Literature | ||
| 20. | ALA1108955 | B | Inhibition of rat recombinant GluA4 receptor expressed in Xenopus oocytes assessed as inhibition of 300 uM kainate-induced current | Rattus norvegicus | 1 | cell-based format | Scientific Literature |
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