# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3789208 | B | Inhibition of recombinant KDM3B (842 to 1761 residues) (unknown origin) expressed in baculovirus infected sf9 cells using biotin-H3K9me as substrate preincubated for 10 mins followed by substrate addition measured after 10 mins by AlphaLisa assay | Homo sapiens | 3 | ALA3784917 | cell-based format | Scientific Literature | |
2. | ALA4022352 | B | Inhibition of KDM3B (unknown origin) at 10 uM | Homo sapiens | 2 | ALA4020786 | single protein format | Scientific Literature | |
3. | ALA4022356 | B | Inhibition of KDM3B (unknown origin) | Homo sapiens | 1 | ALA4020786 | single protein format | Scientific Literature | |
4. | ALA4035839 | B | Inhibition of recombinant human N-terminal FLAG-tagged KDM3B expressed in baculovirus infected Sf9 insect cells using H3K9me1 peptide as substrate after 30 to 45 mins by TR-FRET assay | Homo sapiens | 2 | ALA4033700 | cell-based format | Scientific Literature | |
5. | ALA4193852 | B | Inhibition of KDM3B (unknown origin) using biotinylated H3K9me1 peptide and alpha-ketoglutarate as substrate measured after 20 mins by LANCE TR-FRET assay | Homo sapiens | 1 | ALA4190335 | single protein format | Scientific Literature | |
6. | ALA4427166 | B | Inhibition of KDM3B (unknown origin) | Homo sapiens | 1 | ALA4425149 | single protein format | Scientific Literature | |
7. | ALA4427936 | B | Inhibition of KDM3B (unknown origin) using ARTKQTAR(KMe1)STGGKAPRKQLA -NovaTagPEG-biotin/2-OG as substrate/co-factor by TR-FRET assay | Homo sapiens | 1 | ALA4425189 | single protein format | Scientific Literature | |
8. | ALA4832324 | B | Inhibition of KDM3B (unknown origin) by AlphaLISA assay | Homo sapiens | 1 | ALA4831501 | single protein format | Scientific Literature | |
9. | ALA4836321 | B | Inhibition of KDM3B (unknown origin) by Succinate-Glo assay | Homo sapiens | 1 | ALA4834445 | single protein format | Scientific Literature | |
10. | ALA4836328 | B | Binding affinity to KDM3B (unknown origin) by differential scanning fluorimetry | Homo sapiens | 1 | ALA4834445 | single protein format | Scientific Literature | |
11. | ALA5032407 | B | Inhibition of human N-terminal His6-tagged KDM3B (L882 to S1761 residues) expressed in insect cells using H3K9(Me2) as substrate preincubated for 15 mins followed by substrate addition and measured after 5 mins by Alphascreen assay | Homo sapiens | 13 | ALA5030566 | cell-based format | Scientific Literature | |
12. | ALA5127948 | B | Binding affinity to CM7 sensor chip immobilized full-length KDM3B (unknown origin) expressed in Sf9 insect cells assessed as dissociation constant incubated for 60 secs by SPR analysis | Homo sapiens | 3 | ALA5126529 | cell-based format | Scientific Literature |