# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3991951 | B | Inhibition of human recombinant Glepp-1 catalytic domain using DiFMUP as substrate after 30 mins by fluorescence assay | Homo sapiens | 7 | ALA3991941 | single protein format | Patent Bioactivity Data | |
2. | ALA4374233 | B | Inhibition of recombinant human N-terminal His-tagged PTPRO expressed in bacterial expression system assessed as enzyme residual activity at 2 uM using DiFMUP as substrate preincubated with enzyme for 2.5 hrs prior to substrate addition measured for 1 min by fluorescence based assay | Homo sapiens | 1 | ALA4373652 | assay format | Scientific Literature | |
3. | ALA4374246 | B | Inhibition of recombinant human N-terminal His-tagged PTPRO expressed in bacterial expression system at 2 uM using DiFMUP as substrate preincubated with enzyme and catalase for 2.5 hrs prior to substrate addition measured for 1 min by fluorescence based assay | Homo sapiens | 1 | ALA4373652 | assay format | Scientific Literature | |
4. | ALA4374250 | B | Inhibition of recombinant human N-terminal His-tagged PTPRO expressed in bacterial expression system assessed as rate of product DiFMU formed at 2 uM using DiFMUP as substrate preincubated with enzyme for 2.5 hrs prior to substrate addition measured for 1 min by fluorescence based assay (Rvb = 209.7 nM/sec) | Homo sapiens | 1 | ALA4373652 | assay format | Scientific Literature | |
5. | ALA4768203 | B | Inhibition of GLEEP (unknown origin) | Homo sapiens | 4 | ALA4765268 | single protein format | Scientific Literature | |
6. | ALA5233990 | B | Binding affinity to GLEPP1 (unknown origin) assessed as inhibition constant | Homo sapiens | 1 | ALA5233224 | single protein format | Scientific Literature |