| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4017389 | B | Inhibition of SETb (unknown origin) H3K4 methyltransferase activity using biotinyl-H3 peptide (1 to 21 residues) and using [3H]-S adenosylmethionine as methyl donor up to 100 uM after 1 hr by scintillation counting | Homo sapiens | 1 | ALA4014355 | single protein format | Scientific Literature | |
| 2. | ALA4333233 | B | Inhibition of SETD1B (unknown origin) using SAM as substrate preincubated for 15 mins followed by substrate addition and measured after 1 hr by Alphalisa assay | Homo sapiens | 1 | ALA4330131 | single protein format | Scientific Literature | |
| 3. | ALA4397121 | B | Inhibition of C-terminal GST-tagged human SET1B (1629 to 1923 amino acids) expressed in Escherichia coli using core histone as substrate in presence of WDR5 (22 to 334 amino acids),RbBP5 (1 to 538 amino acids),Ash2L (2 to 534 amino acids),DPY-30 (1 to 99 amino acids) by fluorescence method | Homo sapiens | 1 | ALA4396867 | assay format | Scientific Literature | |
| 4. | ALA4731571 | B | Inhibition of recombinant human N- terminal GST-tagged SET1B (1629 to 1923 residues) expressed in Escherichia coli using core histone as substrate at 10 uM by radiometric HotSpot assay relative to control | Homo sapiens | 1 | ALA4725473 | assay format | Scientific Literature | |
| 5. | ALA5119826 | B | Inhibition of human recombinant N-terminal GST-tagged SET1B (1629 to 1923 residues) expressed in Escherichia coli at 10 uM using GST-GAR as substrate by scintillation/filter plate assay | Homo sapiens | 1 | ALA5113528 | assay format | Scientific Literature | |
| 6. | ALA5119888 | B | Inhibition of human recombinant N-terminal GST-tagged SET1B (1629 to 1923 residues) expressed in Escherichia coli at 50 uM using GST-GAR as substrate by scintillation/filter plate assay relative to control | Homo sapiens | 1 | ALA5113528 | assay format | Scientific Literature | |
| 7. | ALA5129704 | B | Inhibition of N-terminal GST-tagged SET1B (1629 to 1923 residues) (unknown origin) expressed in Escherichia coli at 1 uM using 3H-SAM as a substrate relative to control | Homo sapiens | 1 | ALA5126600 | assay format | Scientific Literature |
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