| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4119040 | B | Binding affinity to PDIA3 in human NCI-H358 cells at 1 uM by mass spectrometry based pull down assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 2. | ALA4257303 | B | Inhibition of ERP57 (unknown origin) assessed as reduction in enzyme-mediated bovine insulin aggregation after 30 mins by turbidimetric assay | Homo sapiens | 9 | single protein format | Patent Bioactivity Data | ||
| 3. | ALA4682778 | B | Inhibition of PDIA3 (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 1 hr and measured by insulin reduction assay | Homo sapiens | 3 | assay format | Scientific Literature | ||
| 4. | ALA4729813 | A | Inhibition of PDIA3 (unknown origin) at 40 uM using bovine insulin as substrate preincubated for 1 hr followed by substrate addition | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 5. | ALA4729843 | A | Inhibition of N-(4-(5,5-Difluoro-1,3,7,9-tetramethyl-5H-4(Gamma4),5(Gamma4)-dipyrrolo[1,2-c:2',1'-f][1,3,2]diazaborinin-10-yl))-N-(2-(4-((6-hydroxybenzo[d]-[1,3]dioxol-5-yl)(piperidin-1-yl)methyl)benzamido)ethyl)-benzamide binding to recombinant PDIA3 (unknown origin) measured after 24 hrs by PAGE analysis | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 6. | ALA5145309 | B | Binding affinity to PDIA3 in human DOHH-2 cells measured after 6 hrs by pull-down assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 7. | ALA5145319 | B | Binding affinity to PDIA3 in human MDA-MB-453 cells measured after 6 hrs by pull-down assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 8. | ALA5145336 | B | Binding affinity to PDIA3 in human DOHH-2 cells at 10 uM measured after 6 hrs in presence of 100 uM PES by pull-down assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 9. | ALA5145353 | B | Binding affinity to PDIA3 in human MDA-MB-453 cells at 10 uM measured after 6 hrs in presence of 100 uM PES by pull-down assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 10. | ALA5145370 | B | Binding affinity to PDIA3 in human DOHH-2 cells by MS analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 11. | ALA5147888 | B | Inhibition of ERp57 (unknown origin) reductase activity assessed as inhibition of PDI/DTT-mediated cleavage of disulfide bond in insulin in the presence of DTT incubated for 40 mins by spectrophotometric analysis | Homo sapiens | 1 | single protein format | Scientific Literature |
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