| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4151497 | B | Inhibition of N-terminal FLAG-tagged human full-length CDK13 (1 to 1512 residues)/N-terminal His-tagged CycK (1 to 580 residues) expressed in Sf9 cells assessed as reduction in ATP-dependent ULight-4E-BP1 (Thr37/Thr46) substrate peptide phosphorylation pre-incubated for 60 mins by LANCE Ultra assay | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 2. | ALA4314617 | B | Inhibition of recombinant full length human CDK13/cyclinK assessed as residual activity at 10 uM using RSRSRSRSRSRSRSR as substrate measured after 120 mins in presence of [gamma33P]ATP by scintillation counting method | Homo sapiens | 1 | protein complex format | Scientific Literature | ||
| 3. | ALA4335009 | B | Inhibition of recombinant full length human CDK13/cyclinK assessed as residual activity at 1 uM using RSRSRSRSRSRSRSR as substrate incubated for 120 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay relative to control | Homo sapiens | 2 | protein complex format | Scientific Literature | ||
| 4. | ALA4336837 | B | Inhibition of recombinant full length human CDK13/cyclinK assessed as residual activity at 10 uM using RSRSRSRSRSRSR as substrate incubated for 40 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay relative to control | Homo sapiens | 1 | protein complex format | Scientific Literature | ||
| 5. | ALA4351792 | B | Inhibition of recombinant full length human CDK13/cyclinK at 10 uM using RSRSRSRSRSRSRSR as substrate measured after 120 mins in presence of [gamma33P]ATP by scintillation counting method | Homo sapiens | 1 | protein complex format | Scientific Literature | ||
| 6. | ALA4377708 | B | Inhibition of human full length recombinant CDK13/cyclinK at 1 uM using RSRSRSRSRSRSRSR as substrate incubated for 120 mins in presence of [gamma-33P]ATP at by radiometric assay relative to control | Homo sapiens | 1 | protein complex format | Scientific Literature | ||
| 7. | ALA4378935 | B | Inhibition of full-length recombinant human CDK13/cyclinK at 10 uM using RSRSRSRSRSRSRSR as substrate after 120 mins by in presence of [gamma33P]ATP by scintillation counting method relative to control | Homo sapiens | 1 | protein complex format | Scientific Literature | ||
| 8. | ALA4379179 | B | Inhibition of recombinant full length human CDK13/cyclinK using RSRSRSRSRSRSR as substrate incubated for 120 mins in presence of [gamma-33ATP] by radiometric scintillation counting analysis | Homo sapiens | 1 | protein complex format | Scientific Literature | ||
| 9. | ALA4387186 | B | Inhibition of tracer 236 binding to human GST/His-tagged CDK13/Cyclin K at 0.1 uM | Homo sapiens | 2 | protein complex format | Scientific Literature | ||
| 10. | ALA4408787 | B | Competitive irreversible inhibition of CDK13/cyclinK (unknown origin) in presence of 1 mM ATP | Homo sapiens | 1 | protein complex format | Scientific Literature | ||
| 11. | ALA4408795 | B | Competitive irreversible inhibition of CDK13/cyclinK (unknown origin) in presence of Km ATP | Homo sapiens | 1 | protein complex format | Scientific Literature | ||
| 12. | ALA4612777 | B | Inhibition of human CDK13/cyclin K using Pol2-CTD as substrate by [gamma-33P]ATP-based radioisotope filter binding assay | Homo sapiens | 1 | protein complex format | Scientific Literature | ||
| 13. | ALA4775151 | B | Inhibition of CDK13/human cyclin K expressed in baculovirus-infected insect cells using pol2 CTD-peptide substrate and [gammaP]ATP by scintillation counting method | 1 | cell-based format | Scientific Literature | |||
| 14. | ALA4828802 | B | Inhibition of human recombinant CDK13/CyclinK assessed as reduction in substrate phosphorylation using His-c-Myc as substrate preincubated with enzyme for 5 mins followed by substrate addition for 15 mins in presence of [gamma 32P-ATP] by radioactive kinase assay | Homo sapiens | 20 | protein complex format | Scientific Literature | ||
| 15. | ALA4830406 | B | Inhibition of human CDK13/cyclin-K incubated for 2 hrs by [gamma-33P]-ATP assay | Homo sapiens | 1 | protein complex format | Scientific Literature | ||
| 16. | ALA4880993 | B | CDK13/cyclinK(h) Eurofins Kinase panel | Homo sapiens | 1 | protein complex format | Donated Chemical Probes - SGC Frankfurt | ||
| 17. | ALA4887251 | B | CDK13/CYCLIN K Invitrogen Lab (UK) kinase screen (BI) | Homo sapiens | 1 | protein complex format | Donated Chemical Probes - SGC Frankfurt | ||
| 18. | ALA4888130 | B | CDK13/cyclinK(h) Millipore kinase panel | Homo sapiens | 1 | protein complex format | Donated Chemical Probes - SGC Frankfurt | ||
| 19. | ALA5041394 | B | Inhibition of CDK13/cyclin-K (unknown origin) | Homo sapiens | 1 | protein complex format | Scientific Literature | ||
| 20. | ALA5104713 | B | Inhibition of recombinant CDK13/Cyclin K (unknown origin) expresssed in baculovirus infected insect cells using peptide substrate incubated for 30 mins in presence of [32P]gamma-ATP by scintillation counter method | Homo sapiens | 1 | assay format | Scientific Literature |
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