# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4264616 | B | Inhibition of recombinant GST-tagged human full length CDK14/cyclin Y (2 to end residues) | Homo sapiens | 1 | ALA4261600 | protein complex format | Scientific Literature | |
2. | ALA4314618 | B | Inhibition of human CDK14/cyclinY assessed as residual activity at 10 uM by radiometric method | Homo sapiens | 1 | ALA4311992 | protein complex format | Scientific Literature | |
3. | ALA4327619 | B | Inhibition of human CDK14/cyclin-Y assessed as residual activity at 1 uM using RB protein as substrate by [gamma-33P]-ATP assay relative to control | Homo sapiens | 2 | ALA4325871 | protein complex format | Scientific Literature | |
4. | ALA4327980 | B | Inhibition of human CDK14/cyclin-Y assessed as residual activity at 100 uM using RB protein as substrate by [gamma-33P]-ATP assay relative to control | Homo sapiens | 1 | ALA4325871 | protein complex format | Scientific Literature | |
5. | ALA4328344 | B | Inhibition of human CDK14/cyclin-Y using RB protein as substrate by [gamma-33P]-ATP assay | Homo sapiens | 1 | ALA4325871 | protein complex format | Scientific Literature | |
6. | ALA4335010 | B | Inhibition of recombinant full length human CDK14/cyclinY assessed as residual activity at 1 uM in presence of [gamma-33ATP] by scintillation counting based radiometry assay relative to control | Homo sapiens | 2 | ALA4334438 | protein complex format | Scientific Literature | |
7. | ALA4336838 | B | Inhibition of recombinant full length human CDK14/cyclinY assessed as residual activity at 10 uM in presence of [gamma-33ATP] by scintillation counting based radiometry assay relative to control | Homo sapiens | 1 | ALA4334471 | protein complex format | Scientific Literature | |
8. | ALA4351794 | B | Inhibition of human CDK14/cyclinY at 10 uM by radiometric method | Homo sapiens | 1 | ALA4350961 | protein complex format | Scientific Literature | |
9. | ALA4366322 | B | Inhibition of human CDK14/cyclin-Y at 100 nM using RB protein as substrate by [gamma-33P]-ATP assay | Homo sapiens | 1 | ALA4364276 | protein complex format | Scientific Literature | |
10. | ALA4377709 | B | Inhibition of human CDK14/cyclinY at 1 uM by radiometric method relative to control | Homo sapiens | 1 | ALA4376814 | protein complex format | Scientific Literature | |
11. | ALA4378934 | B | Inhibition of human CDK14/cyclinY at 10 uM by radiometric assay relative to control | Homo sapiens | 1 | ALA4376829 | protein complex format | Scientific Literature | |
12. | ALA4379180 | B | Inhibition of recombinant full length human CDK14/cyclinY in presence of [gamma-33ATP] by radiometric scintillation counting analysis | Homo sapiens | 1 | ALA4376834 | protein complex format | Scientific Literature | |
13. | ALA4387187 | B | Inhibition of tracer 236 binding to recombinant human GST-tagged CDK14/cyclin Y catalytic domain (CDK14: full length, Cyclin Y: 2 to end) expressed by baculovirus in Sf9 insect cells expression system at 0.1 uM measured after 60 mins by Lanthascreen assay relative to control | Homo sapiens | 2 | ALA4385643 | cell-based format | Scientific Literature | |
14. | ALA4405295 | B | Inhibition of CDK14/Cyclin Y (unknown origin) at 1 uM relative to control | Homo sapiens | 1 | ALA4402587 | protein complex format | Scientific Literature | |
15. | ALA4408790 | B | Competitive irreversible inhibition of CDK14/cyclin Y (unknown origin) in presence of Km ATP | Homo sapiens | 1 | ALA4406837 | protein complex format | Scientific Literature | |
16. | ALA4434176 | B | Inhibition of recombinant GST-tagged human full length CDK14/cyclin Y (2 to end residues) preincubated for 30 mins by Lantha screen eu binding assay | Homo sapiens | 100 | ALA4433236 | protein complex format | Scientific Literature | |
17. | ALA4434179 | B | Covalent binding affinity to GST-tagged human full length CDK14/cyclin Y (2 to end residues) assessed as formation of covalent bond formation at 10:1 M ratio of compound to CDK14/Cyclin Y protein incubated for 3 hrs by MS/MS analysis | Homo sapiens | 2 | ALA4433236 | protein complex format | Scientific Literature | |
18. | ALA4434185 | B | Inhibition of recombinant NanoLuc-tagged CDK14/cyclin Y expressed in human HCT116 cells at 1 uM incubated for 20 to 24 hrs by by NanoBRET assay | Homo sapiens | 1 | ALA4433236 | cell-based format | Scientific Literature | |
19. | ALA4612778 | B | Inhibition of kinase tracer 236 binding to recombinant human N-terminal GST-tagged full-length CDK14/Cyclin Y (2 to end residues) expressed in baculovirus infected Sf9 insect cells measured after 1 hr by LanthaScreen Eu Kinase Binding Assay | Homo sapiens | 1 | ALA4610118 | cell-based format | Scientific Literature | |
20. | ALA4623654 | B | Inhibition of human CDK14/Cyclin Y using RB protein as substrate at 20 uM in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assay relative to control | Homo sapiens | 1 | ALA4622865 | protein complex format | Scientific Literature |