| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4219285 | B | Induction of cereblon/cullin 4A-mediated BRD2 degradation in human RS4:11 cells at 1 nM after 3 hrs in presence of proteosome inhibitor MG-132 by Western blot method | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 2. | ALA4219286 | B | Induction of cereblon/cullin 4A-mediated BRD2 degradation in human RS4:11 cells at 1 nM after 3 hrs in presence of cereblon inhibitor lenalidomide by Western blot method | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 3. | ALA4219291 | B | Induction of cereblon/cullin 4A-mediated BRD2 degradation in human RS4:11 cells at 1 nM after 3 hrs in presence of NAE inhibitor MLN4924 by Western blot method | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 4. | ALA4219295 | B | Induction of cereblon/cullin 4A-mediated BRD2 degradation in human RS4:11 cells at 30 to 1000 nM after 24 hrs by Western blot method | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 5. | ALA4219298 | B | Induction of cereblon/cullin 4A-mediated BRD2 degradation in human RS4:11 cells at 1 nM after 3 hrs in presence of BET inhibitor 4-((3-Cyclopropyl-1-ethyl-1H-pyrazol-5-yl)amino)-7-(3,5-dimethylisoxazol-4-yl)-6-methoxy-N-methyl-9H-pyrimido[4,5-b]-indole-2-carboxamide by Western blot method | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 6. | ALA4219301 | B | Induction of cereblon/cullin 4A-mediated BRD2 degradation in human RS4:11 cells at 30 to 1000 nM after 3 hrs by Western blot method | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 7. | ALA4219303 | B | Induction of cereblon/cullin 4A-mediated BRD2 degradation in human RS4:11 cells at 0.1 nM after 24 hrs by Western blot method | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 8. | ALA4219307 | B | Induction of cereblon/cullin 4A-mediated BRD2 degradation in human RS4:11 cells at 100 to 300 nM after 3 hrs by Western blot method | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 9. | ALA4219309 | B | Induction of cereblon/cullin 4A-mediated BRD2 degradation in human RS4:11 cells at 30 to 300 nM after 3 hrs by Western blot method | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 10. | ALA4219312 | B | Induction of cereblon/cullin 4A-mediated BRD2 degradation in human RS4:11 cells after 3 hrs by Western blot method | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 11. | ALA4219342 | B | Induction of cereblon/cullin 4A-mediated BRD2 degradation in human RS4:11 cells at 3 to 10 nM after 3 hrs by Western blot method | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 12. | ALA4219343 | B | Induction of cereblon/cullin 4A-mediated BRD2 degradation in human RS4:11 cells at 3 to 30 nM after 3 hrs by Western blot method | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 13. | ALA4219347 | B | Induction of cereblon/cullin 4A-mediated BRD2 degradation in human MOLM13 cells after 3 hrs by Western blot method | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 14. | ALA4382975 | B | Protac activity at cereblon/cullin 4A/BRD2 in human RS4:11 cells assessed as BRD2 degradation by Western blot analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 15. | ALA4382978 | B | Protac activity at cereblon/cullin 4A/BRD2 in human RS4:11 cells assessed as BRD2 degradation at 0.1 nM after 3 hrs by Western blot analysis | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 16. | ALA4382999 | B | Protac activity at cereblon/cullin 4A/BRD2 in human RS4:11 cells assessed as BRD2 degradation at 30 to 100 pM after 3 hrs by Western blot analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 17. | ALA4383000 | B | Protac activity at cereblon/cullin 4A/BRD2 in human MV4-11 cells assessed as BRD2 degradation at 30 to 100 pM after 3 hrs by Western blot analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 18. | ALA4383002 | B | Protac activity at cereblon/cullin 4A/BRD2 in human RS4:11 cells assessed as BRD2 degradation at 0.5 nM after 3 hrs by Western blot analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 19. | ALA4383005 | B | Protac activity at cereblon/cullin 4A/BRD2 in human RS4:11 cells assessed as BRD2 degradation at 0.5 nM after 3 hrs in presence of lenalidomide by Western blot analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 20. | ALA4383008 | B | Protac activity at cereblon/cullin 4A/BRD2 in human RS4:11 cells assessed as BRD2 degradation at 0.5 nM after 3 hrs in presence of neddylation inhibitor MLN4924 by Western blot analysis | Homo sapiens | 1 | cell-based format | Scientific Literature |
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