| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5249913 | B | Protac activity at VHL/BRD3 (unknown origin) | Homo sapiens | 1 | protein format | Scientific Literature | ||
| 2. | ALA5249919 | B | Protac activity at VHL/BRD3 in human HeLa cells assessed as degradation of BRD3 incubated for 24 hrs by Western blotting analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 3. | ALA5249927 | B | Protac activity at VHL/BRD3 in HEK293 cells assessed as degradation of BRD3 incubated for 4 hrs by Western blot analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 4. | ALA4190492 | B | Proteolysis targeting chimera activity in human 22Rv1 cells assessed as induction of VHL-mediated delivery of BRD3 for protein degradation by proteasome by measuring drug level causing 50% substrate depletion incubated for 16 hrs by Western blot method | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 5. | ALA4349410 | B | Protac activity against VHL/BRD3 in human VCaP cells assessed as induction of BRD3 protein degradation by reverse phase protein array analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 6. | ALA4349416 | B | Protac activity against VHL/BRD3 (unknown origin) assessed as induction of BRD4 protein degradation by cell based assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 7. | ALA4388594 | B | Protac activity at VHL/BRD3 in human 22Rv1 cells assessed as induction of BRD3 protein degradation incubated for 16 hrs by Western blot analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 8. | ALA5036173 | B | Protac activity at VHL/Brd3 in HEK293 cells assessed as Brd3 degradation after 4 hrs by Western blotting analysis | Homo sapiens | 8 | cell-based format | Scientific Literature | ||
| 9. | ALA5231282 | B | PROTAC activity at BRD3/VHL in human 22Rv1 cells assessed as protein degradation measured after 16 hrs | Homo sapiens | 1 | cell-based format | Scientific Literature |
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