# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA654174 | B | Human calcitonin receptor I1 mediated CRE-luciferase activity in human neuroblastoma cells | Homo sapiens | 13 | ALA1135734 | cell-based format | Scientific Literature | |
2. | ALA654175 | B | Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cells | Homo sapiens | 13 | ALA1135734 | cell-based format | Scientific Literature | |
3. | ALA654176 | B | Affinity for human calcitonin receptor I1 expressed in HEK293 cells relative to [125I]-salmon calcitonin | Homo sapiens | 13 | ALA1135734 | cell-based format | Scientific Literature | |
4. | ALA654537 | B | Human calcitonin receptor I1 mediated CRE-luciferase activity relative to sCT in human neuroblastoma cells | Homo sapiens | 13 | ALA1135734 | cell-based format | Scientific Literature | |
5. | ALA654538 | B | Displacement of [125I]calcitonin from T-47D (human breast cancer) cell membrane expressing human calcitonin receptor | 5 | ALA1133879 | cell-based format | Scientific Literature | ||
6. | ALA1000517 | B | Displacement of [125I]calcitonin from calcitonin receptor in human T47D cells | Homo sapiens | 1 | ALA1156565 | cell-based format | Scientific Literature | |
7. | ALA1909101 | B | DRUGMATRIX: Calcitonin radioligand binding (ligand: [125I] Calcitonin (salmon)) | 871 | ALA1909046 | cell membrane format | DrugMatrix | ||
8. | ALA2040046 | B | Displacement of [125I]calcitonin from human CT receptor expressed in HEK293 cells | Homo sapiens | 1 | ALA2034981 | cell-based format | Scientific Literature | |
9. | ALA3100461 | B | Inhibition of human calcitonin receptor at 10 uM relative to control | Homo sapiens | 1 | ALA3098111 | single protein format | Scientific Literature | |
10. | ALA3624147 | B | Inhibition of human calcitonin receptor at 10 uM relative to control | Homo sapiens | 1 | ALA3621160 | single protein format | Scientific Literature | |
11. | ALA4421024 | F | Agonist activity at human calcitonin receptor expressed in BHK570 cells assessed as increase in intracellular cAMP concentration incubated for 3 hrs in absence of albumin by CRE luciferase reporter gene assay | Homo sapiens | 143 | ALA4420076 | cell-based format | Patent Bioactivity Data | |
12. | ALA4421026 | F | Agonist activity at human calcitonin receptor expressed in BHK570 cells assessed as increase in intracellular cAMP concentration incubated for 3 hrs in presence of 10% FBS by CRE luciferase reporter gene assay | Homo sapiens | 96 | ALA4420076 | cell-based format | Patent Bioactivity Data | |
13. | ALA4421038 | B | Displacement of [125I]-labeled human calcitonin from human calcitonin receptor expressed in BHK tkts13 cell membranes incubated for 1 hr by scintillation proximity assay | Homo sapiens | 39 | ALA4420076 | cell-based format | Patent Bioactivity Data | |
14. | ALA4421040 | B | Displacement of [125I]-labeled rat calcitonin from human calcitonin receptor expressed in BHK tkts13 cell membranes incubated for 1 hr by scintillation proximity assay | Homo sapiens | 39 | ALA4420076 | cell-based format | Patent Bioactivity Data | |
15. | ALA4421073 | B | Displacement of [125I]-labeled human calcitonin from human calcitonin receptor expressed in BHK tkts13 whole cells incubated for 60 mins by scintillation proximity assay | Homo sapiens | 91 | ALA4420076 | cell-based format | Patent Bioactivity Data | |
16. | ALA4880903 | B | Calcitonin Eurofins-Panlabs radioligand binding assay | Homo sapiens | 3 | ALA4507332 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
17. | ALA4883325 | B | PRESTO-Tango GPCRome screening (CALCRb) | 1 | ALA4507309 | single protein format | Donated Chemical Probes - SGC Frankfurt |