# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4482362 | B | Inhibition of human recombinant MEST T579B (2 to 335 amino acids) expressed in Sf9 cell membranes assessed as reduction in glycerol 3-phosphate acyltransferase activity at 200 uM using [3H]-glycerol 3-phosphate and palmitoyl CoA incubated for 60 mins by scintillation counting assay relative to control | Homo sapiens | 1 | ALA4482303 | cell-based format | Patent Bioactivity Data | |
2. | ALA4482363 | B | Inhibition of human recombinant MEST T579B (2 to 335 amino acids) expressed in Sf9 cell membranes assessed as reduction in glycerol 3-phosphate acyltransferase activity at 100 uM using [3H]-glycerol 3-phosphate and palmitoyl CoA incubated for 60 mins by scintillation counting assay relative to control | Homo sapiens | 1 | ALA4482303 | cell-based format | Patent Bioactivity Data | |
3. | ALA4482364 | B | Inhibition of human recombinant MEST T579B (2 to 335 amino acids) expressed in Sf9 cell membranes assessed as reduction in glycerol 3-phosphate acyltransferase activity at 30 uM using [3H]-glycerol 3-phosphate and palmitoyl CoA incubated for 60 mins by scintillation counting assay relative to control | Homo sapiens | 1 | ALA4482303 | cell-based format | Patent Bioactivity Data | |
4. | ALA4482365 | B | Inhibition of human recombinant MEST T579B (2 to 335 amino acids) expressed in Sf9 cell membranes assessed as reduction in glycerol 3-phosphate acyltransferase activity at 10 uM using [3H]-glycerol 3-phosphate and palmitoyl CoA incubated for 60 mins by scintillation counting assay relative to control | Homo sapiens | 2 | ALA4482303 | cell-based format | Patent Bioactivity Data | |
5. | ALA4482366 | B | Inhibition of human recombinant MEST T579B (2 to 335 amino acids) expressed in Sf9 cell membranes assessed as reduction in glycerol 3-phosphate acyltransferase activity at 3 uM using [3H]-glycerol 3-phosphate and palmitoyl CoA incubated for 60 mins by scintillation counting assay relative to control | Homo sapiens | 2 | ALA4482303 | cell-based format | Patent Bioactivity Data | |
6. | ALA4482367 | B | Inhibition of human recombinant MEST T579B (2 to 335 amino acids) expressed in Sf9 cell membranes assessed as reduction in glycerol 3-phosphate acyltransferase activity at 1 uM using [3H]-glycerol 3-phosphate and palmitoyl CoA incubated for 60 mins by scintillation counting assay relative to control | Homo sapiens | 2 | ALA4482303 | cell-based format | Patent Bioactivity Data | |
7. | ALA4482368 | B | Inhibition of human recombinant MEST T579B (2 to 335 amino acids) expressed in Sf9 cell membranes assessed as reduction in glycerol 3-phosphate acyltransferase activity at 0.3 uM using [3H]-glycerol 3-phosphate and palmitoyl CoA incubated for 60 mins by scintillation counting assay relative to control | Homo sapiens | 2 | ALA4482303 | cell-based format | Patent Bioactivity Data | |
8. | ALA4482369 | B | Inhibition of human recombinant MEST T579B (2 to 335 amino acids) expressed in Sf9 cell membranes assessed as reduction in glycerol 3-phosphate acyltransferase activity using [3H]-glycerol 3-phosphate and palmitoyl CoA incubated for 60 mins by scintillation counting assay | Homo sapiens | 2 | ALA4482303 | cell-based format | Patent Bioactivity Data | |
9. | ALA4482370 | B | Inhibition of human recombinant MEST T579B (2 to 335 amino acids) expressed in Sf9 cell membranes assessed as reduction in glycerol 3-phosphate acyltransferase activity at 0.1 uM using [3H]-glycerol 3-phosphate and palmitoyl CoA incubated for 60 mins by scintillation counting assay relative to control | Homo sapiens | 1 | ALA4482303 | cell-based format | Patent Bioactivity Data | |
10. | ALA4482371 | B | Inhibition of human recombinant MEST T579B (2 to 335 amino acids) expressed in Sf9 cell membranes assessed as reduction in glycerol 3-phosphate acyltransferase activity at 0.03 uM using [3H]-glycerol 3-phosphate and palmitoyl CoA incubated for 60 mins by scintillation counting assay relative to control | Homo sapiens | 1 | ALA4482303 | cell-based format | Patent Bioactivity Data | |
11. | ALA4482390 | B | Inhibition of human recombinant MEST T580B (11 to 335 amino acids) expressed in Sf9 cell membranes assessed as reduction in glycerol 3-phosphate acyltransferase activity at 10 uM using [3H]-glycerol 3-phosphate and palmitoyl CoA incubated for 60 mins by scintillation counting assay relative to control | Homo sapiens | 1 | ALA4482303 | cell-based format | Patent Bioactivity Data | |
12. | ALA4482391 | B | Inhibition of human recombinant MEST T580B (11 to 335 amino acids) expressed in Sf9 cell membranes assessed as reduction in glycerol 3-phosphate acyltransferase activity at 3 uM using [3H]-glycerol 3-phosphate and palmitoyl CoA incubated for 60 mins by scintillation counting assay relative to control | Homo sapiens | 1 | ALA4482303 | cell-based format | Patent Bioactivity Data | |
13. | ALA4482392 | B | Inhibition of human recombinant MEST T580B (11 to 335 amino acids) expressed in Sf9 cell membranes assessed as reduction in glycerol 3-phosphate acyltransferase activity at 1 uM using [3H]-glycerol 3-phosphate and palmitoyl CoA incubated for 60 mins by scintillation counting assay relative to control | Homo sapiens | 1 | ALA4482303 | cell-based format | Patent Bioactivity Data | |
14. | ALA4482393 | B | Inhibition of human recombinant MEST T580B (11 to 335 amino acids) expressed in Sf9 cell membranes assessed as reduction in glycerol 3-phosphate acyltransferase activity at 0.3 uM using [3H]-glycerol 3-phosphate and palmitoyl CoA incubated for 60 mins by scintillation counting assay relative to control | Homo sapiens | 1 | ALA4482303 | cell-based format | Patent Bioactivity Data | |
15. | ALA4482394 | B | Inhibition of human recombinant MEST T580B (11 to 335 amino acids) expressed in Sf9 cell membranes assessed as reduction in glycerol 3-phosphate acyltransferase activity at 0.1 uM using [3H]-glycerol 3-phosphate and palmitoyl CoA incubated for 60 mins by scintillation counting assay relative to control | Homo sapiens | 1 | ALA4482303 | cell-based format | Patent Bioactivity Data | |
16. | ALA4482395 | B | Inhibition of human recombinant MEST T580B (11 to 335 amino acids) expressed in Sf9 cell membranes assessed as reduction in glycerol 3-phosphate acyltransferase activity at 0.03 uM using [3H]-glycerol 3-phosphate and palmitoyl CoA incubated for 60 mins by scintillation counting assay relative to control | Homo sapiens | 1 | ALA4482303 | cell-based format | Patent Bioactivity Data | |
17. | ALA4482397 | B | Inhibition of human recombinant MEST T579B (2 to 335 amino acids) expressed in Sf9 cell membranes assessed as reduction in glycerol 3-phosphate acyltransferase activity at 1 mM using [3H]-glycerol 3-phosphate and palmitoyl CoA in presence of 30 ug MEST enzyme incubated for 1 hr by scintillation counting assay relative to control | Homo sapiens | 1 | ALA4482303 | cell-based format | Patent Bioactivity Data | |
18. | ALA4482398 | B | Inhibition of human recombinant MEST T580B (11 to 335 amino acids) expressed in Sf9 cell membranes assessed as reduction in glycerol 3-phosphate acyltransferase activity at 1 mM using [3H]-glycerol 3-phosphate and palmitoyl CoA in presence of 30 ug MEST enzyme incubated for 1 hr by scintillation counting assay relative to control | Homo sapiens | 1 | ALA4482303 | cell-based format | Patent Bioactivity Data | |
19. | ALA4482400 | B | Inhibition of human recombinant MEST T579B (2 to 335 amino acids) expressed in Sf9 cell membranes assessed as reduction in glycerol 3-phosphate acyltransferase activity at 1 mM using [3H]-glycerol 3-phosphate and palmitoyl CoA in presence of 10 ug MEST enzyme incubated for 1 hr by scintillation counting assay relative to control | Homo sapiens | 1 | ALA4482303 | cell-based format | Patent Bioactivity Data | |
20. | ALA4482401 | B | Inhibition of human recombinant MEST T580B (11 to 335 amino acids) expressed in Sf9 cell membranes assessed as reduction in glycerol 3-phosphate acyltransferase activity at 1 mM using [3H]-glycerol 3-phosphate and palmitoyl CoA in presence of 10 ug MEST enzyme incubated for 1 hr by scintillation counting assay relative to control | Homo sapiens | 1 | ALA4482303 | cell-based format | Patent Bioactivity Data |