# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4327806 | B | Inhibition of human OSR1 assessed as residual activity at 1 uM using RRHYYYDTHTNTYYLRTFGHNTRR as substrate by [gamma-33P]-ATP assay relative to control | Homo sapiens | 2 | ALA4325871 | single protein format | Scientific Literature | |
2. | ALA4328170 | B | Inhibition of human OSR1 assessed as residual activity at 100 uM using RRHYYYDTHTNTYYLRTFGHNTRR as substrate by [gamma-33P]-ATP assay relative to control | Homo sapiens | 1 | ALA4325871 | single protein format | Scientific Literature | |
3. | ALA4328534 | B | Inhibition of human OSR1 using RRHYYYDTHTNTYYLRTFGHNTRR as substrate by [gamma-33P]-ATP assay | Homo sapiens | 1 | ALA4325871 | single protein format | Scientific Literature | |
4. | ALA4352474 | B | Inhibition of human OSR1 at 10 uM using RRHYYYDTHTNTYYLRTFGHNTRR as substrate in presence of [gamma-33P]-ATP | Homo sapiens | 1 | ALA4350963 | single protein format | Scientific Literature | |
5. | ALA4674268 | B | Inhibition of human OSR1 using RRHYYYDTHTNTYYLRTFGHNTRR as substrate assessed as residual activity at 1 uM by [gamma-33P]-ATP assay relative to control | Homo sapiens | 2 | ALA4673210 | single protein format | Scientific Literature | |
6. | ALA4720621 | B | Inhibition of human OSR1 using RRHYYYDTHTNTYYLRTFGHNTRR as substrate by [gamma-33P]-ATP assay | Homo sapiens | 1 | ALA4715818 | single protein format | Scientific Literature | |
7. | ALA4720968 | B | Inhibition of human OSR1 assessed as residual activity using RRHYYYDTHTNTYYLRTFGHNTRR as substrate at 1 uM by [gamma-33P]-ATP assay relative to control | Homo sapiens | 1 | ALA4715818 | single protein format | Scientific Literature | |
8. | ALA4721476 | B | Inhibition of wild-type human full length OSR1 (M1 to S527 residues) expressed in mammalian expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4715821 | assay format | Scientific Literature | |
9. | ALA4805063 | B | Inhibition of human OSR1 assessed as percent of control at 2000 nM by KINOMEscan assay relative to control | Homo sapiens | 1 | ALA4804282 | single protein format | Patent Bioactivity Data | |
10. | ALA4805651 | B | Inhibition of human OSR1 assessed as percent of control at 1000 nM by KINOMEscan assay relative to control | Homo sapiens | 1 | ALA4804283 | single protein format | Patent Bioactivity Data | |
11. | ALA4806108 | B | Inhibition of DNA-tagged human OSR1 assessed as percent of control at 50000 nM by qPCR analysis relative to control | Homo sapiens | 1 | ALA4804284 | single protein format | Patent Bioactivity Data | |
12. | ALA4806668 | B | Inhibition of human OSR1 assessed as percent of control at 2000 nM by KINOMEscan assay relative to control | Homo sapiens | 1 | ALA4804286 | single protein format | Patent Bioactivity Data | |
13. | ALA5058303 | B | Inhibition of OSR1 (unknown origin) at 1 uM | Homo sapiens | 1 | ALA5055685 | single protein format | Scientific Literature | |
14. | ALA5231871 | B | Inhibition of human full-length GST-tagged OSR1 T185E mutant expressed in Escherichia coli BL21 (DE3) incubated for 30 min in presence of ATP by HTS based ADP-Glo kinase assay | Homo sapiens | 1 | ALA5230131 | assay format | Scientific Literature |