| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4324380 | B | Inhibition of NTMT1 (unknown origin) assessed as enzyme activity at 3.7 uM using GPKRIA peptide as substrate preincubated for 10 mins in presence of AdoMet followed by susbtrate addition by fluorescence based SAHH enzyme coupled assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 2. | ALA4324388 | B | Inhibition of NTMT1 (unknown origin) assessed as enzyme activity at 11 uM using GPKRIA peptide as substrate preincubated for 10 mins in presence of AdoMet followed by susbtrate addition by fluorescence based SAHH enzyme coupled assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 3. | ALA4324396 | B | Inhibition of NTMT1 (unknown origin) assessed as enzyme activity at 33 uM using GPKRIA peptide as substrate preincubated for 10 mins in presence of AdoMet followed by susbtrate addition by fluorescence based SAHH enzyme coupled assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 4. | ALA4324404 | B | Inhibition of NTMT1 (unknown origin) assessed as enzyme activity at 100 uM using GPKRIA peptide as substrate preincubated for 10 mins in presence of AdoMet followed by susbtrate addition by fluorescence based SAHH enzyme coupled assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 5. | ALA4324412 | B | Inhibition of NTMT1 (unknown origin) using GPKRIA peptide as substrate preincubated for 10 mins in presence of AdoMet followed by susbtrate addition by fluorescence based SAHH enzyme coupled assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 6. | ALA4392203 | B | Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cells using GPKRIA as substrate preincubated for 10 mins in presence of SAM followed by substrate addition by fluorescence assay | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 7. | ALA4392204 | B | Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cells at 10 uM using GPKRIA as substrate preincubated for 10 mins in presence of SAM followed by substrate addition by fluorescence assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 8. | ALA4392205 | B | Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cells assessed as reduction in GPKRIA trimethylation at 50 nM preincubated for 10 mins in presence of SAM followed by GPKRIA addition and measured after 20 mins by MALDI TOF-MS analysis relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 9. | ALA4392206 | B | Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cells assessed as reduction in GPKRIA trimethylation at 100 nM preincubated for 10 mins in presence of SAM followed by GPKRIA addition and measured after 20 mins by MALDI TOF-MS analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 10. | ALA4392207 | B | Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cells assessed as reduction in GPKRIA di-methylation at 100 nM preincubated for 10 mins in presence of SAM followed by GPKRIA addition and measured after 20 mins by MALDI TOF-MS analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 11. | ALA4392208 | B | Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cells preincubated for 10 mins in presence of SAM followed by GPKRIA addition and measured after 20 mins by MALDI TOF-MS analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 12. | ALA4392209 | B | Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cells assessed as residual enzyme activity at 3.3 uM using GPKRIA as substrate preincubated for 10 mins in presence of SAM followed by substrate addition by fluorescence assay relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 13. | ALA4392210 | B | Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cells assessed as residual enzyme activity at 10 uM using GPKRIA as substrate preincubated for 10 mins in presence of SAM followed by substrate addition by fluorescence assay relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 14. | ALA4392247 | B | Bi-substrate inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cells using varying levels of GPKRIA as substrate preincubated for 10 mins in presence of varying levels of SAM followed by substrate addition by fluorescence assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 15. | ALA4392248 | B | Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cells using peptide substrate in presence of SAM by fluorescence assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 16. | ALA4392249 | B | Inhibition of recombinant human full-length His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cells using SPKRIAKRRS as substrate in presence of SAM by fluorescence assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 17. | ALA4621543 | B | Inhibition of NTMT1 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 18. | ALA4621544 | B | Substrate activity at NTMT1 (unknown origin) assessed as compound methylation at 10 uM incubated overnight by MALDI-MS methylation assay | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 19. | ALA4621545 | B | Inhibition of NTMT1 (unknown origin) pre-incubated for 10 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence assay | Homo sapiens | 8 | single protein format | Scientific Literature | ||
| 20. | ALA4621546 | B | Inhibition of NTMT1 (unknown origin) pre-incubated for 10 mins before GPKRIA peptide substrate addition and measured after 20 mins by MALDI-MS methylation assay | Homo sapiens | 1 | single protein format | Scientific Literature |
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