| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4370954 | B | Protac activity against VHL/cullin2/ERalpha in human MCF7 cells assessed as ERalpha degradation by measuring ER protein/GADPH ratio at 1 nM after 4 hrs by Western blot analysis relative to control | Homo sapiens | 36 | cell-based format | Scientific Literature | ||
| 2. | ALA4370955 | B | Protac activity against VHL/cullin2/ERalpha in human MCF7 cells assessed as ERalpha degradation by measuring ER protein/GADPH ratio at 10 nM after 4 hrs by Western blot analysis relative to control | Homo sapiens | 36 | cell-based format | Scientific Literature | ||
| 3. | ALA4370956 | B | Protac activity against VHL/cullin2/ERalpha in human MCF7 cells assessed as ERalpha degradation by measuring ER protein/GADPH ratio at 100 nM after 4 hrs by Western blot analysis relative to control | Homo sapiens | 36 | cell-based format | Scientific Literature | ||
| 4. | ALA4370957 | B | Protac activity against VHL/cullin2/ERalpha in human MCF7 cells assessed as ERalpha degradation by measuring ER protein/GADPH ratio at 1000 nM after 4 hrs by Western blot analysis relative to control | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 5. | ALA4370959 | B | Protac activity against VHL/cullin2/ERalpha in human MCF7 cells assessed as ERalpha degradation after 4 hrs by Western blot analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 6. | ALA4370960 | B | Protac activity against VHL/cullin2/ERalpha in human MCF7 cells assessed as ERalpha degradation by measuring ER protein/GAPDH ratio at 0.03 nM after 4 hrs by Western blot analysis relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 7. | ALA4370961 | B | Protac activity against VHL/cullin2/ERalpha in human MCF7 cells assessed as ERalpha degradation by measuring ER protein/GAPDH ratio at 0.3 nM after 4 hrs by Western blot analysis relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 8. | ALA4370962 | B | Protac activity against VHL/cullin2/ERalpha in human MCF7 cells assessed as ERalpha degradation by measuring ER protein/GAPDH ratio at 0.6 nM after 4 hrs by Western blot analysis relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 9. | ALA4370963 | B | Protac activity against VHL/cullin2/ERalpha in human MCF7 cells assessed as ERalpha degradation by measuring ER protein/GAPDH ratio at 5 nM after 4 hrs by Western blot analysis relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 10. | ALA4370964 | B | Protac activity against VHL/cullin2/ERalpha in human MCF7 cells assessed as ERalpha degradation by measuring ER protein/GAPDH ratio at 30 nM after 4 hrs by Western blot analysis relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 11. | ALA4370965 | B | Protac activity against VHL/cullin2/ERalpha in human MCF7 cells assessed as ERalpha degradation by measuring ER protein/GAPDH ratio at 300 nM after 4 hrs by Western blot analysis relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 12. | ALA4370966 | B | Protac activity against VHL/cullin2/ERalpha in human T47D cells assessed as ERalpha degradation by measuring ER protein/GAPDH ratio at 0.03 nM after 4 hrs by Western blot analysis relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 13. | ALA4370967 | B | Protac activity against VHL/cullin2/ERalpha in human T47D cells assessed as ERalpha degradation by measuring ER protein/GAPDH ratio at 0.1 nM after 4 hrs by Western blot analysis relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 14. | ALA4370968 | B | Protac activity against VHL/cullin2/ERalpha in human T47D cells assessed as ERalpha degradation by measuring ER protein/GAPDH ratio at 0.3 nM after 4 hrs by Western blot analysis relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 15. | ALA4370969 | B | Protac activity against VHL/cullin2/ERalpha in human T47D cells assessed as ERalpha degradation by measuring ER protein/GAPDH ratio at 0.6 nM after 4 hrs by Western blot analysis relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 16. | ALA4370970 | B | Protac activity against VHL/cullin2/ERalpha in human T47D cells assessed as ERalpha degradation by measuring ER protein/GAPDH ratio at 1 nM after 4 hrs by Western blot analysis relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 17. | ALA4370971 | B | Protac activity against VHL/cullin2/ERalpha in human T47D cells assessed as ERalpha degradation by measuring ER protein/GAPDH ratio at 5 nM after 4 hrs by Western blot analysis relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 18. | ALA4370972 | B | Protac activity against VHL/cullin2/ERalpha in human T47D cells assessed as ERalpha degradation by measuring ER protein/GAPDH ratio at 10 nM after 4 hrs by Western blot analysis relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 19. | ALA4370973 | B | Protac activity against VHL/cullin2/ERalpha in human T47D cells assessed as ERalpha degradation by measuring ER protein/GAPDH ratio at 30 nM after 4 hrs by Western blot analysis relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 20. | ALA4370974 | B | Protac activity against VHL/cullin2/ERalpha in human T47D cells assessed as ERalpha degradation by measuring ER protein/GAPDH ratio at 100 nM after 4 hrs by Western blot analysis relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature |
The page will load shortly, Thanks for your patience!