| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4830744 | F | Agonist activity at human GPR27 expressed in HEK293 cells co-expressing FnLArrb2.GPR27V2LFc assessed as induction of beta-arrestin recruitment incubated for 10 mins measured followed by addition of D-luciferin by firefly-luciferase complementation assay | Homo sapiens | 31 | cell-based format | Scientific Literature | ||
| 2. | ALA4830745 | F | Agonist activity at human GPR27 expressed in HEK293 cells co-expressing FnLArrb2.GPR27V2LFc assessed as maximal induction of beta-arrestin recruitment incubated for 10 mins measured followed by addition of D-luciferin by firefly-luciferase complementation assay relative to control | Homo sapiens | 31 | cell-based format | Scientific Literature | ||
| 3. | ALA4830747 | F | Agonist activity at human GPR27 expressed in HEK293 cells assessed as induction of beta-arrestin recruitment pretreated with substrate for 45 mins followed by compound addition and measured for 40 mins by NanoLuc luciferase complementation assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 4. | ALA4883443 | B | PRESTO-Tango GPCRome screening (GPR27) | 1 | single protein format | Donated Chemical Probes - SGC Frankfurt |
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