| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1837770 | B | Inhibition of human PKACgamma in HL60 cells lysate at 10 uM using post probe-labeling by LC-MS/MS analysis relative to control | Homo sapiens | 5 | ALA1833925 | cell-based format | Scientific Literature | |
| 2. | ALA3630925 | B | Inhibition of PKAcgamma (unknown origin) at 10 uM after 120 mins P33 radiolabeled kinase activity assay | Homo sapiens | 3 | ALA3627608 | single protein format | Scientific Literature | |
| 3. | ALA3748053 | B | Inhibition of human PKAcgamma using [KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK] as substrate | Homo sapiens | 1 | ALA3745707 | single protein format | Scientific Literature | |
| 4. | ALA3991838 | B | Kinobeads (epsilon), multiple immobilized ATP-competitive broad spectrum kinase inhibitors, used to assess residual binding of ~300 proteins simultaneously from cell lysate in the presence of a compound. Quantitative readout performed by mass spectrometry. | Homo sapiens | 200 | ALA3991601 | subcellular format | Kuster lab chemical proteomics drug profiling | |
| 5. | ALA4322837 | B | Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged PRKACG (unknown origin) expressed in baculovirus infected Sf9 insect cells incubated for 1 hr by TR-FRET assay | Homo sapiens | 2 | ALA4321812 | cell-based format | Scientific Literature | |
| 6. | ALA4327832 | B | Inhibition of human PKAcg assessed as residual activity at 1 uM using KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK as substrate by [gamma-33P]-ATP assay relative to control | Homo sapiens | 2 | ALA4325871 | single protein format | Scientific Literature | |
| 7. | ALA4328196 | B | Inhibition of human PKAcg assessed as residual activity at 100 uM using KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK as substrate by [gamma-33P]-ATP assay relative to control | Homo sapiens | 1 | ALA4325871 | single protein format | Scientific Literature | |
| 8. | ALA4328560 | B | Inhibition of human PKAcg using KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK as substrate by [gamma-33P]-ATP assay | Homo sapiens | 1 | ALA4325871 | single protein format | Scientific Literature | |
| 9. | ALA4352499 | B | Inhibition of human PKAcg at 10 uM using KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK as substrate in presence of [gamma-33P]-ATP | Homo sapiens | 1 | ALA4350963 | single protein format | Scientific Literature | |
| 10. | ALA4366544 | B | Inhibition of human PKAcg at 100 nM using KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK as substrate by [gamma-33P]-ATP assay | Homo sapiens | 1 | ALA4364276 | single protein format | Scientific Literature | |
| 11. | ALA4405516 | B | Inhibition of PRKAC-gamma (unknown origin) at 1 uM relative to control | Homo sapiens | 1 | ALA4402587 | single protein format | Scientific Literature | |
| 12. | ALA4606503 | A | Inhibition of recombinant human full-length N-terminal GST-tagged PKAcgamma expressed in baculovirus infected Sf9 insect cells at 1 uM by Lanthascreen assay relative to control | Homo sapiens | 1 | ALA4602732 | cell-based format | Scientific Literature | |
| 13. | ALA4674242 | B | Inhibition of human PKAcg using KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK as substrate assessed as residual activity at 1 uM by [gamma-33P]-ATP assay relative to control | Homo sapiens | 2 | ALA4673210 | single protein format | Scientific Literature | |
| 14. | ALA4720597 | B | Inhibition of human PKAcg using KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK as substrate by [gamma-33P]-ATP assay | Homo sapiens | 1 | ALA4715818 | single protein format | Scientific Literature | |
| 15. | ALA4720942 | B | Inhibition of human PKAcg assessed as residual activity using KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK as substrate at 1 uM by [gamma-33P]-ATP assay relative to control | Homo sapiens | 1 | ALA4715818 | single protein format | Scientific Literature | |
| 16. | ALA4721500 | B | Inhibition of PKAcg (unknown origin) assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4715821 | single protein format | Scientific Literature | |
| 17. | ALA4884823 | B | PKAgamma(PRCGLGY1) Takeda global kinase panel | Homo sapiens | 1 | ALA4507327 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
| 18. | ALA4885114 | B | PKAgamma(PRCGLGY1) Takeda global kinase panel | Homo sapiens | 1 | ALA4507326 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
| 19. | ALA4885400 | B | PKAgamma(PRCGLGY1) Takeda global kinase panel | Homo sapiens | 1 | ALA4507327 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
| 20. | ALA4887315 | B | PRKACG (PRKAC GAM Invitrogen Lab (UK) kinase screen (BI) | Homo sapiens | 1 | ALA4800722 | single protein format | Donated Chemical Probes - SGC Frankfurt |
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