# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA860800 | B | Average Binding Constant for MYLK2; NA=Not Active at 10 uM | Homo sapiens | 20 | ALA1144455 | single protein format | Scientific Literature | |
2. | ALA990530 | B | Inhibition of MYLK2 | 1 | ALA1149823 | single protein format | Scientific Literature | ||
3. | ALA987207 | B | Inhibition of MYLK2 at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
4. | ALA1061160 | B | Binding constant for MYLK2 kinase domain | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
5. | ALA1048289 | B | Inhibition of MYLK2 assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
6. | ALA1043342 | B | Residual activity of MYLK2 at 0.1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
7. | ALA1041154 | B | Residual activity of MYLK2 at 1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
8. | ALA1050307 | B | Residual activity of MYLK2 at 10 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
9. | ALA1100972 | B | Inhibition of MYLK2 at 10 uM | 2 | ALA1154277 | single protein format | Scientific Literature | ||
10. | ALA1105927 | B | Inhibition of skeletal MLCK at 5 uM | 1 | ALA1154316 | single protein format | Scientific Literature | ||
11. | ALA1166585 | B | Inhibition of MYLK2 at 1 uM | 10 | ALA1165965 | single protein format | Scientific Literature | ||
12. | ALA1174933 | B | Inhibition of MYLK2 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
13. | ALA1244226 | B | Inhibition of MYLK2 at 1 uM after 60 mins by FRET assay in presence of 100 uM ATP | 7 | ALA1240340 | single protein format | Scientific Literature | ||
14. | ALA1244531 | B | Binding affinity to MYLK2 | 7 | ALA1240346 | single protein format | Scientific Literature | ||
15. | ALA1249592 | B | Inhibition of His-tagged human SkMLCK expressed in Escherichia coli at 20 uM | Homo sapiens | 1 | ALA1240295 | assay format | Scientific Literature | |
16. | ALA1249784 | B | Inhibition of His-tagged human SkMLCK expressed in Escherichia coli at 1 uM | Homo sapiens | 1 | ALA1240295 | assay format | Scientific Literature | |
17. | ALA1252497 | B | Inhibition of MYLK2 at 1 uM in presence of 100 uM ATP by Select Screen kinase assay relative to untreated control | 3 | ALA1250448 | single protein format | Scientific Literature | ||
18. | ALA1633369 | B | Inhibition of MYLK2 at 10 uM | 1 | ALA1629532 | single protein format | Scientific Literature | ||
19. | ALA1646789 | B | Inhibition of MYLK2 at 1 uM | 1 | ALA1641460 | single protein format | Scientific Literature | ||
20. | ALA1646933 | B | Inhibition of MYLK2 at 10 uM | 1 | ALA1641460 | single protein format | Scientific Literature |