# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA673366 | Binding | Inhibition of Dual-specificity tyrosine-phosphorylation regulated kinase 1A at 10 uM | Homo sapiens | 3 | ALA1136207 | single protein format | Scientific Literature | |
2. | ALA673367 | Binding | Inhibition of Dual-specificity tyrosine-phosphorylation regulated kinase 1A at 10 uM | Homo sapiens | 1 | ALA1136207 | single protein format | Scientific Literature | |
3. | ALA1292141 | Binding | Inhibition of human DYRK1A | Homo sapiens | 1 | ALA1287713 | single protein format | Scientific Literature | |
4. | ALA1057274 | Binding | Inhibition of human recombinant GST-fusion DYRK1A expressed in Escherichia coli | Homo sapiens | 14 | ALA1153477 | assay format | Scientific Literature | |
5. | ALA1052085 | Binding | Percentage DYRK1A activity remaining in the presence of 0.01uM inhibitor | Homo sapiens | 3 | ALA1150976 | single protein format | Scientific Literature | |
6. | ALA1062880 | Binding | Inhibition of DYRK1A in the presence of 50uM ATP | Homo sapiens | 1 | ALA1150976 | single protein format | Scientific Literature | |
7. | ALA1063743 | Binding | Percentage DYRK1A activity remaining in the presence of 10uM inhibitor | Homo sapiens | 24 | ALA1150976 | single protein format | Scientific Literature | |
8. | ALA1051344 | Binding | Inhibition of DYRK1a | 1 | ALA1150975 | single protein format | Scientific Literature | ||
9. | ALA1051376 | Binding | Percentage DYRK1A activity remaining in the presence of 0.1uM inhibitor | Homo sapiens | 7 | ALA1150976 | single protein format | Scientific Literature | |
10. | ALA1051377 | Binding | Percentage DYRK1A activity remaining in the presence of 25uM inhibitor | Homo sapiens | 2 | ALA1150976 | single protein format | Scientific Literature | |
11. | ALA1060112 | Binding | Percentage DYRK1A activity remaining in the presence of 2uM inhibitor | Homo sapiens | 1 | ALA1150976 | single protein format | Scientific Literature | |
12. | ALA1060231 | Binding | Percent residual DYRK1a activity in the presence of 10uM inhibitor | 3 | ALA1150975 | single protein format | Scientific Literature | ||
13. | ALA1062005 | Binding | Percentage DYRK1A activity remaining in the presence of 1uM inhibitor | Homo sapiens | 33 | ALA1150976 | single protein format | Scientific Literature | |
14. | ALA1062006 | Binding | Percentage DYRK1A activity remaining in the presence of 3uM inhibitor | Homo sapiens | 1 | ALA1150976 | single protein format | Scientific Literature | |
15. | ALA1041352 | Binding | Inhibition of DYRK1A at 1 uM | 1 | ALA1154622 | single protein format | Scientific Literature | ||
16. | ALA1041498 | Binding | Inhibition of DYRK1R | 1 | ALA1154675 | single protein format | Scientific Literature | ||
17. | ALA1043730 | Binding | Inhibition of DYRK1A assessed as residual activity at 10 uM by Cherenkov counting relative to control in presence of 50 uM ATP | 2 | ALA1155278 | single protein format | Scientific Literature | ||
18. | ALA1049892 | Binding | Inhibition of DYRK1A assessed as residual activity at 0.1 uM by Cherenkov counting relative to control in presence of 50 uM ATP | 2 | ALA1155278 | single protein format | Scientific Literature | ||
19. | ALA1049460 | Binding | Residual activity of DYRK1A at 0.1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
20. | ALA1037123 | Binding | Residual activity of DYRK1A at 1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature |