| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA651140 | F | Activity for beta 3-adrenoceptor was assessed from effect on stimulation of lipolysis in rat adipocytes. | 2 | ALA1128729 | cell-based format | Scientific Literature | ||
| 2. | ALA651142 | F | In vitro beta adrenergic receptor activity against beta-3 adrenergic receptor in rat epididymal fat pads by stimulation of glycerol release from adipocytes. | 1 | ALA1125527 | tissue-based format | Scientific Literature | ||
| 3. | ALA651143 | F | In vitro beta-adrenergic activity against beta-3 adrenergic receptor in rat epididymal fat pads by stimulation of glycerol release from adipocytes. | 3 | ALA1125527 | tissue-based format | Scientific Literature | ||
| 4. | ALA651144 | F | Effective dose for contraction of reserpine-pretreated rat vas deferens | 1 | ALA1128729 | tissue-based format | Scientific Literature | ||
| 5. | ALA651145 | B | Inhibition of beta-3 adrenergic receptor GDP binding in rat brown adipose tissue on oral administration relative to isoprenaline | Rattus norvegicus | 11 | ALA1126035 | tissue-based format | Scientific Literature | |
| 6. | ALA651146 | B | Dose necessary to produce 50% of the isoprenaline effect to inhibit GDP binding to beta-3 adrenergic receptor in brown adipose tissue (BAT mitochondria) of rats after subcutaneous administration. | 28 | ALA1126035 | mitochondrion format | Scientific Literature | ||
| 7. | ALA651147 | B | Dose necessary to produce 50% of the isoprenaline effect to inhibit GDP binding to beta-3 adrenergic receptor in brown adipose tissue(BAT mitochondria) of rats after subcutaneous administration; not active | 1 | ALA1126035 | mitochondrion format | Scientific Literature | ||
| 8. | ALA651900 | B | Dose of the compound (peroral administration) to inhibit GDP binding against Beta-3 adrenergic receptor in brown adipose tissue(BAT mitochondria) of rats. [Dose necessary to produce 50% of the isoprenaline effect] | 1 | ALA1126292 | mitochondrion format | Scientific Literature | ||
| 9. | ALA655027 | B | Dose of the compound (peroral administration) to inhibit GDP binding against Beta-3 adrenergic receptor in brown adipose tissue(BAT mitochondria) of rats; Not tested | 1 | ALA1126292 | mitochondrion format | Scientific Literature | ||
| 10. | ALA654485 | B | Inhibition of GDP binding against beta-3 adrenergic receptor in brown adipose tissue (BAT) mitochondria of rats after peroral administration (Dose necessary to produce 50% of the isoprenaline effect). | 49 | ALA1126292 | mitochondrion format | Scientific Literature | ||
| 11. | ALA654486 | B | Dose of the compound (peroral administration) to inhibit GDP binding against beta-3 adrenergic receptor in brown adipose tissue(BAT mitochondria) of rats. [Dose necessary to produce 50% of the isoprenaline effect]; Not tested | 2 | ALA1126292 | mitochondrion format | Scientific Literature | ||
| 12. | ALA654487 | B | Peroral dose induction of beta-3 adrenergic receptor mediated GDP binding to mitochondria of rat BAT | Rattus norvegicus | 14 | ALA1126292 | single protein format | Scientific Literature | |
| 13. | ALA856081 | F | Agonistic activity against Beta-3 adrenergic receptor in rat colon | 1 | ALA1128085 | assay format | Scientific Literature | ||
| 14. | ALA818916 | F | Effective dose required for beta-3-adrenergic activity against free fatty acid (FFA) in rat plasma | Rattus norvegicus | 9 | ALA1131783 | cell-free format | Scientific Literature | |
| 15. | ALA818917 | F | Beta-3-adrenergic activity measured by percent response against free fatty acid (FFA) in rat plasma at a dosage of 0.1 mg/kg | 92 | ALA1131783 | organism-based format | Scientific Literature | ||
| 16. | ALA818918 | F | Compound was evaluated for the beta-3-adrenergic activity by measuring % response against free fatty acid (FFA) in rat plasma at a dosage of 0.1 mg/kg | 1 | ALA1131783 | organism-based format | Scientific Literature | ||
| 17. | ALA819430 | F | Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret detrusor | 19 | ALA1134410 | assay format | Scientific Literature | ||
| 18. | ALA819431 | F | Agonistic activity towards beta-3 adrenoceptor. EC50, the mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret detrusor | 1 | ALA1134410 | assay format | Scientific Literature | ||
| 19. | ALA819432 | F | Activity compared to that observed following forskolin (10e -5). | 20 | ALA1134410 | assay format | Scientific Literature | ||
| 20. | ALA840720 | F | Ratio of the dose raising the rat heart rate to 500bpm, to ED50 for inhibition of GDP binding to beta-3 adrenergic receptor | Rattus norvegicus | 21 | ALA1126035 | tissue-based format | Scientific Literature |
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