| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA709029 | F | Inhibition of MEK-1 Kinase phosphorylation in LoVo cells | 1 | ALA1146624 | cell-based format | Scientific Literature | ||
| 2. | ALA734036 | B | Inhibition of Mitogen activated protein kinase kinase kinase 1 at 1 uM | 3 | ALA1149171 | single protein format | Scientific Literature | ||
| 3. | ALA729501 | B | Inhibitory potency against mitogen activated protein kinase kinase kinase 1 at 10 uM | 1 | ALA1147629 | single protein format | Scientific Literature | ||
| 4. | ALA880238 | B | Inhibitory concentration against Mitogen-activated protein kinase kinase kinase 1 (MEKK1) | Homo sapiens | 1 | ALA1141086 | single protein format | Scientific Literature | |
| 5. | ALA934583 | B | Inhibition of MEKK | 1 | ALA1142440 | single protein format | Scientific Literature | ||
| 6. | ALA1031537 | B | Inhibition of MEKK1 | 1 | ALA1152750 | single protein format | Scientific Literature | ||
| 7. | ALA1041531 | B | Inhibition of C-terminal FLAG-tagged MEKK1 by [gamma-33-P]ATP based assay | 2 | ALA1154165 | single protein format | Scientific Literature | ||
| 8. | ALA1045292 | B | Inhibition of MAPK3K1 at 3 uM | 1 | ALA1156783 | single protein format | Scientific Literature | ||
| 9. | ALA1116699 | B | Inhibition of MAP3K1 at 5 uM | 1 | ALA1154316 | single protein format | Scientific Literature | ||
| 10. | ALA1166055 | B | Inhibition of MAP3K1 at 1 uM | 6 | ALA1165965 | single protein format | Scientific Literature | ||
| 11. | ALA1174888 | B | Inhibition of MAP3K1 at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
| 12. | ALA1244369 | B | Inhibition of MAP3K1 | 1 | ALA1240341 | single protein format | Scientific Literature | ||
| 13. | ALA1244489 | B | Binding affinity to MAP3K1 | 7 | ALA1240346 | single protein format | Scientific Literature | ||
| 14. | ALA1826612 | B | Activity of MAP3K1 kinase at 1 uM | 1 | ALA1821651 | single protein format | Scientific Literature | ||
| 15. | ALA1825843 | B | Inhibition of MEKK1 assessed as residual activity at 10 uM by radioactivity assay in presence of 20 uM ATP | 1 | ALA1821675 | single protein format | Scientific Literature | ||
| 16. | ALA1908723 | B | Binding constant for MAP3K1 kinase domain | 72 | ALA1908390 | single protein format | Scientific Literature | ||
| 17. | ALA1924899 | B | Inhibition of C-terminus flag-tagged MEKK1 expressed in baculovirus infected insect cells using [gamma33P]ATP as substrate after 60 mins by scintillation counting | 1 | ALA1921673 | cell-based format | Scientific Literature | ||
| 18. | ALA1943315 | B | Inhibition of human MAP3K1 in HL-60 cells lysate assessed as reduction of labeling of acyl-phosphate ATP probe at 100 nM | Homo sapiens | 4 | ALA1938230 | cell-based format | Scientific Literature | |
| 19. | ALA2014953 | B | Inhibition of MAP3K1 at 10 uM | 1 | ALA2010722 | single protein format | Scientific Literature | ||
| 20. | ALA2015155 | B | Inhibition of MEKK1 assessed as residual activity at 10 uM relative to control | 1 | ALA2010643 | single protein format | Scientific Literature |
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