# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA658286 | B | Binding affinity to cloned human CRF1 receptor expressed in CHO cells using [125I]o-CRF as radioligand at 10 uM concentration; In activie | 1 | cell-based format | Scientific Literature | |||
2. | ALA666036 | F | Effective concentration to stimulate the human corticotropin releasing factor receptor using agonist-stimulated adenylate cyclase assay | 1 | assay format | Scientific Literature | |||
3. | ALA666037 | B | Binding affinity for transfected human Corticotropin releasing factor receptor expressed in HEK 293E cells using [125I]TYR-oCRH as the displaced radioligand | 25 | cell-based format | Scientific Literature | |||
4. | ALA666038 | B | Compound was tested for the binding affinity to human corticotropin releasing factor receptor | 1 | single protein format | Scientific Literature | |||
5. | ALA666039 | B | Compound was tested for the inhibition of binding of the radioligand, [125 I-Tyr0]-CRF to rat cerebral cortex membrane | 1 | tissue-based format | Scientific Literature | |||
6. | ALA666690 | F | Effective dose against CRF stimulated cAMP production in CHO cells expressing human Corticotropin releasing factor receptor 1 | 2 | cell-based format | Scientific Literature | |||
7. | ALA666691 | F | Effective dose against human Corticotropin releasing factor receptor 1 stimulated ACTH release from primary rat anterior pituitary cell cultures | 2 | cell-based format | Scientific Literature | |||
8. | ALA666692 | F | Inhibition of recombinant corticotropin releasing factor receptor 1 assayed using nonselective [125I]-labeled agonist [Tyr0,Glu1,Nle17]-sauvagine | 28 | assay format | Scientific Literature | |||
9. | ALA663518 | B | Displacement of [125I]-TYR-ovine CRH from cloned human corticotropin releasing factor receptor 1 expressed in 293 EBNA cells | 36 | cell-based format | Scientific Literature | |||
10. | ALA663519 | B | Inhibition of [125I]CRH binding to human Corticotropin releasing factor receptor 1. | 18 | single protein format | Scientific Literature | |||
11. | ALA663520 | F | Antagonistic activity for Corticotropin releasing factor receptor 1 | 14 | assay format | Scientific Literature | |||
12. | ALA663521 | B | Displacement of [125I]-tyrosine-ovine-CRF from human Corticotropin releasing factor receptor 1 | Homo sapiens | 14 | single protein format | Scientific Literature | ||
13. | ALA663522 | B | Binding affinity against human Corticotropin releasing factor receptor 1 | 63 | single protein format | Scientific Literature | |||
14. | ALA663523 | B | Binding affinity against human Corticotropin releasing factor receptor 1; Not determined | 2 | single protein format | Scientific Literature | |||
15. | ALA881289 | B | Binding affinity against human Corticotropin releasing factor receptor 1 expressed in HEK 293E cells using [125I]TYR-oCRH | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
16. | ALA666465 | B | Binding affinity to the cloned human corticotropin releasing factor receptor 1 | 28 | single protein format | Scientific Literature | |||
17. | ALA666466 | B | Binding affinity of compound towards human Corticotropin releasing factor receptor 1 | 3 | single protein format | Scientific Literature | |||
18. | ALA666467 | B | Binding affinity towards human corticotropin releasing factor (h-CRF1) receptor | 39 | single protein format | Scientific Literature | |||
19. | ALA666468 | B | Binding affinity of compound towards human corticotropin releasing factor (h-CRF1) receptor showed a 2-fold activity in racemic mixture | 1 | single protein format | Scientific Literature | |||
20. | ALA666469 | B | Binding affinity of compound towards human corticotropin releasing factor (h-CRF1) receptor showed a 2-fold activity in racemic mixture; inactive | 1 | single protein format | Scientific Literature |