# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA642866 | B | Inhibitory activity against adrenergic alpha-receptor transmission, its effect being blocked by phentolamine | Felis catus | 1 | ALA1121518 | single protein format | Scientific Literature | |
2. | ALA640031 | F | Efficacy against alpha 1A adrenoceptor in human expressed as phenylephrine response at the dose of 40 uM | 26 | ALA1134725 | assay format | Scientific Literature | ||
3. | ALA640032 | F | Agonist potency against cloned human alpha 1A adrenoceptor expressed in rat-1 fibroblasts. | 29 | ALA1134725 | assay format | Scientific Literature | ||
4. | ALA642029 | B | Binding affinity was determined on human cloned Alpha-1A adrenoceptor | 8 | ALA1134307 | single protein format | Scientific Literature | ||
5. | ALA646166 | B | Displacement of [125I]HEAT from human Alpha-1C adrenergic receptor expressed in CHO cells | Homo sapiens | 13 | ALA1132031 | cell-based format | Scientific Literature | |
6. | ALA646167 | B | Binding affinity towards human Alpha-1C adrenergic receptor by the displacement of [3H]prazosin | 7 | ALA1127980 | single protein format | Scientific Literature | ||
7. | ALA646331 | B | Compound was evaluated for binding affinity against Alpha-1C adrenergic receptor using radioligand binding assay | 1 | ALA1153669 | single protein format | Scientific Literature | ||
8. | ALA644964 | B | The binding affinity towards Alpha-1C adrenergic receptor in the COS cell line. | 8 | ALA1132568 | cell-based format | Scientific Literature | ||
9. | ALA641525 | B | Binding affinity towards Alpha1A dog adrenergic receptors, using [125I]HEAT as radioligand. | Canis lupus familiaris | 1 | ALA1133777 | single protein format | Scientific Literature | |
10. | ALA640541 | B | Binding affinity towards Alpha1A human adrenergic receptors, using [125I]-HEAT as radioligand. | 1 | ALA1133777 | single protein format | Scientific Literature | ||
11. | ALA641224 | F | Activation of human alpha-1A adrenergic receptor expressed in rat-1 fibroblasts; expressed as a percent of the maximal effect of the phenylephrine | 21 | ALA1134991 | assay format | Scientific Literature | ||
12. | ALA641225 | F | Activation of human alpha-1A adrenergic receptor expressed in rat-1 fibroblasts | 23 | ALA1134991 | assay format | Scientific Literature | ||
13. | ALA641226 | B | In vitro binding affinity against cloned human alpha-1A-adrenoceptor receptors expressed in rat-1 fibroblasts | 8 | ALA1134991 | assay format | Scientific Literature | ||
14. | ALA648627 | B | In vitro affinity for Alpha-1a adrenergic receptor in isolated dog aorta tissue preparations was determined by functional assay | Canis lupus familiaris | 1 | ALA1131394 | tissue-based format | Scientific Literature | |
15. | ALA648628 | B | In vitro affinity for Alpha-1a adrenergic receptor in isolated dog prostate tissue preparations was determined by functional assay | Canis lupus familiaris | 1 | ALA1131394 | tissue-based format | Scientific Literature | |
16. | ALA648629 | B | Compound was evaluated for its affinity for Alpha-1a adrenergic receptor in dog aorta preparations | Canis lupus familiaris | 2 | ALA1131394 | tissue-based format | Scientific Literature | |
17. | ALA648630 | B | Compound was evaluated for its affinity for Alpha-1a adrenergic receptor in dog prostate tissue preparations | Canis lupus familiaris | 2 | ALA1131394 | tissue-based format | Scientific Literature | |
18. | ALA648631 | B | Ability to displace beta ([125I]-iodo-4-hydroxyphenyl)-ethylamino methyl tetralone from human cloned Alpha-1a adrenergic receptor stably expressed in Chinese Hamster Ovary (CHO) cells | Homo sapiens | 11 | ALA1131394 | cell-based format | Scientific Literature | |
19. | ALA648783 | B | Ability to displace beta ([125I]-iodo-4-hydroxyphenyl)-ethylaminomethyl tetralone from human Alpha-1a adrenergic receptor stably expressed in Chinese Hamster Ovary (CHO) cells | 1 | ALA1131394 | cell-based format | Scientific Literature | ||
20. | ALA648784 | B | Ability to displace beta ([125I]-iodo-4-hydroxyphenyl)-ethylaminomethyl tetralone from human cloned Alpha-1a adrenergic receptor stably expressed in CHO cells | 2 | ALA1131394 | cell-based format | Scientific Literature |