| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1825339 | F | Agonist activity at rat recombinant TRPV2 receptor expressed in HEK293 cells assessed as stimulation of intracellular calcium level using Fluo4-AM dye based fluorimetric assay relative to 4 uM ionomycin | Rattus norvegicus | 2 | cell-based format | Scientific Literature | ||
| 2. | ALA1825340 | F | Agonist activity at rat recombinant TRPV2 receptor expressed in HEK293 cells assessed as stimulation of intracellular calcium level using Fluo4-AM dye based fluorimetric assay | Rattus norvegicus | 2 | cell-based format | Scientific Literature | ||
| 3. | ALA1825341 | F | Antagonist activity at rat recombinant TRPV2 receptor expressed in HEK293 cells assessed as inhibition of 3 uM lysophosphatidylcholine-induced stimulation of intracellular calcium level using Fluo4-AM dye based fluorimetric assay | Rattus norvegicus | 2 | cell-based format | Scientific Literature | ||
| 4. | ALA1176319 | F | Antagonist activity at rat TRPV2 receptor | Rattus norvegicus | 1 | assay format | Scientific Literature | ||
| 5. | ALA4143894 | B | Agonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluorescence assay | Rattus norvegicus | 2 | cell-based format | Scientific Literature | ||
| 6. | ALA4235225 | B | Agonist activity at rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence assay relative to ionomycin | Rattus norvegicus | 6 | cell-based format | Scientific Literature | ||
| 7. | ALA4235226 | B | Agonist activity at rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence assay | Rattus norvegicus | 6 | cell-based format | Scientific Literature | ||
| 8. | ALA4235227 | B | Antagonist activity at rat TRPV2 expressed in HEK293 cells assessed as inhibition of LPC-induced increase in intracellular calcium level pretreated for 5 mins followed by LPC addition by Fluo-4-AM dye based fluorescence assay | Rattus norvegicus | 6 | cell-based format | Scientific Literature | ||
| 9. | ALA4236713 | B | Antagonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as inhibition of LPC-induced Ca2+ levels preincubated for 5 mins followed by agonist addition by Fuo-4-AM based spectrofluorimetry | Rattus norvegicus | 50 | cell-based format | Scientific Literature | ||
| 10. | ALA4236714 | B | Antagonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as inhibition of CBD-induced Ca2+ levels preincubated for 5 mins followed by agonist addition by Fuo-4-AM based spectrofluorimetry | Rattus norvegicus | 50 | cell-based format | Scientific Literature | ||
| 11. | ALA4236715 | B | Non-competitive antagonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as inhibition of LPC-induced Ca2+ levels preincubated for 5 mins followed by agonist addition by Fuo-4-AM dependent spectrofluorimetry based Schild analysis | Rattus norvegicus | 3 | cell-based format | Scientific Literature | ||
| 12. | ALA4236716 | B | Non-competitive antagonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as inhibition of CBD-induced Ca2+ levels preincubated for 5 mins followed by agonist addition by Fuo-4-AM dependent spectrofluorimetry based Schild analysis | Rattus norvegicus | 3 | cell-based format | Scientific Literature | ||
| 13. | ALA4377085 | B | Inhibition of YFP-tagged rat TRPV2 expressed in HEK293 cells assessed as reduction in calcium level by fluo-4 dye based fluorescence assay | Rattus norvegicus | 1 | cell-based format | Scientific Literature | ||
| 14. | ALA4478090 | B | Antagonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as inhibition of LPC-induced intracellular calcium accumulation preincubated for 5 mins followed by LPC addition by Fluo-4-AM probe-based spectrofluorimetric assay | Rattus norvegicus | 4 | cell-based format | Scientific Literature | ||
| 15. | ALA4478096 | B | Antagonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as inhibition of LPC-induced intracellular calcium accumulation up to 10 uM preincubated for 5 mins followed by LPC addition by Fluo-4-AM probe-based spectrofluorimetric assay | Rattus norvegicus | 4 | cell-based format | Scientific Literature | ||
| 16. | ALA4675876 | B | Antagonist activity at rat TRPV2 expressed in HEK293 cells assessed as inhibition of LPC-induced Ca2+ response preincubated for 5 mins followed by LPC addition by Fluo-4AM dye based fluorescence assay | Rattus norvegicus | 2 | cell-based format | Scientific Literature | ||
| 17. | ALA4675877 | B | Agonist activity at rat TRPV2 stably transfected in HEK293 cells assessed as increase in calcium influx in presence of ionomycin by Fluo-4-AM dye based spectrofluorimetric method | Rattus norvegicus | 2 | cell-based format | Scientific Literature | ||
| 18. | ALA4675878 | B | Agonist activity at rat TRPV2 stably transfected in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based spectrofluorimetric method relative to ionomycin | Rattus norvegicus | 2 | cell-based format | Scientific Literature |
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