# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA684582 | Binding | Inhibition against human granzyme B | 17 | ALA1134869 | single protein format | Scientific Literature | ||
2. | ALA684583 | Binding | Compound was tested for its inhibition against human granzyme B; Not active | 3 | ALA1134869 | single protein format | Scientific Literature | ||
3. | ALA684584 | Binding | Tested for inhibition of Granzyme B by the compound; ND = Not determined | 3 | ALA1149106 | single protein format | Scientific Literature | ||
4. | ALA684585 | Binding | Tested for inhibition of granzyme B by the compound | 4 | ALA1149106 | single protein format | Scientific Literature | ||
5. | ALA684735 | Binding | Tested for inhibition of granzyme B by the compound; ND = Not determined | 1 | ALA1149106 | single protein format | Scientific Literature | ||
6. | ALA684736 | Binding | Tested for inhibition of granzyme B by the compound; NI = No Inhibition | 1 | ALA1149106 | single protein format | Scientific Literature | ||
7. | ALA684737 | Binding | Tested for inhibition of granzyme B; ND = Not determined | 1 | ALA1149106 | single protein format | Scientific Literature | ||
8. | ALA684738 | Binding | Apparent second-order rate constant was determined by the inhibition of Granzyme B with the compound at the concentration 150 mM; ki/Ki(1/M*s), Not inhibited | 2 | ALA1130861 | single protein format | Scientific Literature | ||
9. | ALA1218388 | Binding | Inhibition of granzyme B-mediated aggregation at 30 uM after 30 mins by spectrophotometry in absence of Triton X-100 | 2 | ALA1212726 | single protein format | Scientific Literature | ||
10. | ALA1218389 | Binding | Inhibition of granzyme B-mediated aggregation at 30 uM after 30 mins by spectrophotometry in presence of Triton X-100 | 2 | ALA1212726 | single protein format | Scientific Literature | ||
11. | ALA948945 | Binding | Inhibition of granzyme B | 3 | ALA1143211 | single protein format | Scientific Literature | ||
12. | ALA2340441 | Binding | Inhibition of Granzyme B (unknown origin) using Ac-IEPD-AMC substrate incubated for 15 mins prior to substrate addition measured for 2 hrs | Homo sapiens | 1 | ALA2331221 | single protein format | Scientific Literature | |
13. | ALA2339097 | Binding | Inhibition of Granzyme B (unknown origin) using Ac-IEPD-AMC substrate assessed as residual activity at 10 uM incubated for 15 mins prior to substrate addition measured for 2 hrs | Homo sapiens | 1 | ALA2331221 | single protein format | Scientific Literature | |
14. | ALA4038153 | Binding | Inhibition of recombinant human Granzyme B (21 to 247 residues) using fluorogenic Ac-IEPD-pNA peptide as substrate by fluorescence based assay | Homo sapiens | 3 | ALA4033799 | single protein format | Scientific Literature | |
15. | ALA4344608 | Binding | Substrate activity at Granzyme B (unknown origin) expressed in Pichia pastoris incubated for 30 mins by fluorescence based assay | Homo sapiens | 1 | ALA4342470 | assay format | Scientific Literature | |
16. | ALA4344612 | Binding | Substrate activity at Granzyme B (unknown origin) expressed in Pichia pastoris assessed as compound hydrolysis at 200 uM incubated for 30 mins by fluorescence based assay relative to control | Homo sapiens | 3 | ALA4342470 | assay format | Scientific Literature | |
17. | ALA4344615 | Binding | Inhibition of Granzyme B (unknown origin) expressed in Pichia pastoris using GrBref substrate by spectrofluorometry relative to control | Homo sapiens | 2 | ALA4342470 | assay format | Scientific Literature |